SCHEMBL11248973

SCHEMBL11248973

O=C(O)c1ccc(NCC(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)F)cc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.47
EPHX2 P34913 3/20 0.40
FNTA P49354 1/20 0.38
FNTB P49356 1/20 0.38
MITF O75030 1/20 0.38
SRD5A2 P31213 2/20 0.38
FAAH O00519 1/20 0.38
TP53 P04637 1/20 0.38
TSHR P16473 1/20 0.38
ALDH1A1 P00352 2/20 0.36
NR1H4 Q96RI1 1/20 0.36
CA1 P00915 2/20 0.36
POLB P06746 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35
RXRG P48443 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11255583 0.80 PDK1 (0.54) CA2TP53TSHRALDH1A1CA1
SCHEMBL10507363 0.80 ALDH1A1 (0.43) CA2ALDH1A1CA1
SCHEMBL1542761 0.80 EPHX2 (0.46) EPHX2FNTAFNTBMITFSRD5A2
Perflubutane SCHEMBL28930534 0.77 TSHR (0.63) CA2SRD5A2TP53TSHRALDH1A1
SCHEMBL5406972 0.77 CA2 (0.38) CA2ALDH1A1CA1
SCHEMBL11317356 0.76 CA2 (0.36) CA2ALDH1A1CA1
SCHEMBL11247397 0.75 PRSS1 (0.43) CA2EPHX2CA1POLB
SCHEMBL26983179 0.75 FFAR1 (0.50) CA2EPHX2SRD5A2ALDH1A1NR1H4
SCHEMBL19964254 0.73 EPHX2 (0.50) CA2EPHX2FNTAFNTBMITF
SCHEMBL17501646 0.72 ALDH1A1 (0.46) CA2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4310545-A Hypolipidemic and antiatherosclerotic 4-(polyfluoroalkylamino) phenyl compounds AMERICAN CYANAMID COMPANY (US) 1982-01-12 US claimed
US-4318914-A Hypolipidemic and antiatherosclerotic 4-(polyfluoro-alkylamino)phenyl compounds AMERICAN CYANAMID COMPANY (US) 1982-03-09 US disclosed
US-4310545-A Hypolipidemic and antiatherosclerotic 4-(polyfluoroalkylamino) phenyl compounds AMERICAN CYANAMID COMPANY (US) 1982-01-12 US disclosed
US-4305959-A Hypolipidemic and antiatherosclerotic 4-(polyfluoro-alkylamino)phenyl compounds AMERICAN CYANAMID COMPANY (US) 1981-12-15 US disclosed
US-4205085-A Hypolipidemic and antiatherosclerotic 4-(polyfluoroalkylamino)phenyl compounds AMERICAN CYANAMID COMPANY (US) 1980-05-27 US disclosed
EP-0003663-A2 Amino-substituted phenyl and heteroaryl compounds, process for their preparation and pharmaceutical compositions containing them AMERICAN CYANAMID COMPANY (US) 1979-08-22 EP disclosed