SCHEMBL11255583

SCHEMBL11255583

CCOC(=O)c1ccc(NCC(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)F)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.54
PDK2 Q15119 1/20 0.54
PDK3 Q15120 1/20 0.54
PDK4 Q16654 1/20 0.54
MAPT P10636 5/20 0.49
MEN1 O00255 4/20 0.49
KMT2A Q03164 4/20 0.49
CASP3 P42574 1/20 0.49
TRPV1 Q8NER1 1/20 0.49
SENP7 Q9BQF6 1/20 0.49
HPGD P15428 2/20 0.48
RECQL P46063 1/20 0.48
RAB9A P51151 7/20 0.47
NPC1 O15118 4/20 0.47
ALDH1A1 P00352 3/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
TSHR P16473 2/20 0.47
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
SMN1; SMN2 Q16637 6/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13985099 0.83 PDK1 (0.58) PDK1PDK2PDK3PDK4MAPT
SCHEMBL11248973 0.80 CA2 (0.47) MEN1KMT2AALDH1A1TSHRCA1
SCHEMBL13410336 0.76 CA1 (0.51) PDK1PDK2PDK3PDK4MAPT
SCHEMBL11261250 0.75 PDK1 (0.53) PDK1PDK2PDK3PDK4MAPT
Perflubutane SCHEMBL28622862 0.75 SMN1; SMN2 (0.56) PDK1PDK2PDK3PDK4MAPT
SCHEMBL13444627 0.75 LMNA (0.61) MAPTMEN1KMT2ACASP3TRPV1
SCHEMBL7101006 0.75 MAPT (0.60) MAPTMEN1KMT2ACASP3TRPV1
SCHEMBL3083718 0.75 HPGD (0.63) MAPTMEN1KMT2ACASP3TRPV1
SCHEMBL9804183 0.75 HPGD (0.63) MAPTMEN1KMT2ACASP3TRPV1
SCHEMBL5067501 0.73 LMNA (0.67) PDK1PDK2PDK3PDK4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4318914-A Hypolipidemic and antiatherosclerotic 4-(polyfluoro-alkylamino)phenyl compounds AMERICAN CYANAMID COMPANY (US) 1982-03-09 US disclosed
US-4310545-A Hypolipidemic and antiatherosclerotic 4-(polyfluoroalkylamino) phenyl compounds AMERICAN CYANAMID COMPANY (US) 1982-01-12 US disclosed
US-4305959-A Hypolipidemic and antiatherosclerotic 4-(polyfluoro-alkylamino)phenyl compounds AMERICAN CYANAMID COMPANY (US) 1981-12-15 US disclosed
US-4205085-A Hypolipidemic and antiatherosclerotic 4-(polyfluoroalkylamino)phenyl compounds AMERICAN CYANAMID COMPANY (US) 1980-05-27 US disclosed
EP-0003663-A2 Amino-substituted phenyl and heteroaryl compounds, process for their preparation and pharmaceutical compositions containing them AMERICAN CYANAMID COMPANY (US) 1979-08-22 EP disclosed