SCHEMBL11249151

SCHEMBL11249151

COc1ccc2c(c1)CCn1cc(-c3ccc(-c4ccccc4)cc3)nc1-2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.49
LMNA P02545 4/20 0.49
NPC1 O15118 4/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
KDM4E B2RXH2 3/20 0.49
ALDH1A1 P00352 3/20 0.49
MAPT P10636 3/20 0.49
THRB P10828 1/20 0.49
HPGD P15428 1/20 0.49
ALDH1A3 P47895 2/20 0.48
WDR5 P61964 3/20 0.46
GAA P10253 1/20 0.45
KMT2A Q03164 1/20 0.45
PDE10A Q9Y233 3/20 0.43
PDE7A Q13946 1/20 0.43
PDE3A Q14432 1/20 0.43
ESR1 P03372 1/20 0.42
HTT P42858 2/20 0.42
ADORA1 P30542 1/20 0.42
EBP Q15125 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11256134 0.91 ALDH1A3 (0.48) RAB9ALMNANPC1SMN1; SMN2KDM4E
SCHEMBL11262715 0.86 PDE10A (0.56) RAB9ALMNANPC1SMN1; SMN2KDM4E
SCHEMBL11247542 0.82 NPC1 (0.52) RAB9ALMNANPC1SMN1; SMN2KDM4E
SCHEMBL11251615 0.81 ALDH1A1 (0.68) RAB9ALMNANPC1SMN1; SMN2KDM4E
SCHEMBL11257591 0.81 RAB9A (0.61) RAB9ALMNANPC1SMN1; SMN2KDM4E
SCHEMBL11249432 0.78 NPC1 (0.52) RAB9ALMNANPC1SMN1; SMN2KDM4E
SCHEMBL8182056 0.75 WDR5 (0.41) RAB9ALMNANPC1SMN1; SMN2WDR5
SCHEMBL11263541 0.75 NPC1 (0.59) RAB9ALMNANPC1SMN1; SMN2KDM4E
SCHEMBL11246624 0.75 NPC1 (0.49) RAB9ALMNANPC1SMN1; SMN2KDM4E
SCHEMBL11252704 0.74 NPC1 (0.65) RAB9ALMNANPC1SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4313950-A Antireproductive tricyclic ortho-fused nitrogen containing compounds GRUPPO LEPETIT S.P.A. (IT) 1982-02-02 US disclosed
US-4275066-A 1,2,4-TRIAZOLO(5.1A)ISOINDOZE, TRIAZOLO(5.1A) ISOQUINOLINE OR 1,2,4,-TRIAZOLO (5.1A)(2) BENZAZEPINE CONTRACEPTIVES GRUPPO LEPETIT S.P.A. (IT) 1981-06-23 US disclosed