SCHEMBL11249174

SCHEMBL11249174

Cc1nn(-c2ccccc2)c(C)c1CC(N)=O

nearest known ligand 0.69

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.69
RAB9A P51151 2/20 0.69
TSHR P16473 1/20 0.63
P2RX7 Q99572 15/20 0.62
MEN1 O00255 1/20 0.57
KMT2A Q03164 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1195590 0.88 NPC1 (0.73) NPC1RAB9ATSHRP2RX7MEN1
SCHEMBL11255334 0.82 TSHR (0.76) NPC1RAB9ATSHRP2RX7MEN1
SCHEMBL8573833 0.82 NPC1 (0.54) NPC1RAB9ATSHRP2RX7MEN1
SCHEMBL11243796 0.81 PDE4D (0.63) NPC1RAB9ATSHRP2RX7MEN1
SCHEMBL11250369 0.80 NPC1 (0.59) NPC1RAB9ATSHRP2RX7MEN1
SCHEMBL8512906 0.79 NPC1 (0.62) NPC1RAB9ATSHRP2RX7MEN1
SCHEMBL11250227 0.79 MEN1 (0.66) NPC1RAB9ATSHRP2RX7MEN1
SCHEMBL1194306 0.78 P2RX7 (0.78) P2RX7
SCHEMBL12770960 0.77 MEN1 (0.68) NPC1RAB9ATSHRP2RX7MEN1
SCHEMBL11539322 0.77 RAB9A (0.58) NPC1RAB9ATSHRP2RX7MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4325962-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIDYRETICS BYK-GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1982-04-20 US disclosed
US-4146721-A ANALGESICS, ANTIINFLAMMATORY AGENTS AND ANTIPYRETICS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1979-03-27 US disclosed