SCHEMBL11249784

SCHEMBL11249784

CCCCOc1ccc(CC(=O)CCn2ccnc2)cc1

nearest known ligand 0.65

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 8/20 0.65
CYP19A1 P11511 2/20 0.60
SMN1; SMN2 Q16637 3/20 0.57
LMNA P02545 2/20 0.57
PLA2G4A P47712 1/20 0.56
KDM4E B2RXH2 2/20 0.56
HTT P42858 2/20 0.56
MAPK1 P28482 1/20 0.56
GAA P10253 1/20 0.55
ALDH1A1 P00352 1/20 0.55
QPCT Q16769 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11255655 0.86 TBXAS1 (0.56) TBXAS1CYP19A1PLA2G4A
SCHEMBL11261566 0.86 KDM4E (0.63) TBXAS1SMN1; SMN2LMNAPLA2G4AKDM4E
SCHEMBL11240600 0.85 CYP19A1 (0.60) TBXAS1CYP19A1KDM4EGAAALDH1A1
SCHEMBL11260419 0.84 TBXAS1 (0.59) TBXAS1
SCHEMBL11259784 0.83 TBXAS1 (0.55) TBXAS1SMN1; SMN2KDM4EALDH1A1QPCT
SCHEMBL11178893 0.81 PLA2G4A (0.72) TBXAS1CYP19A1SMN1; SMN2LMNAPLA2G4A
SCHEMBL11236348 0.81 CYP19A1 (0.56) TBXAS1CYP19A1ALDH1A1QPCT
SCHEMBL11238134 0.81 MEN1 (0.59) TBXAS1CYP19A1KDM4EGAAALDH1A1
SCHEMBL11265550 0.81 TBXAS1 (0.57) TBXAS1CYP19A1PLA2G4A
SCHEMBL11242023 0.79 KMT2A (0.53) TBXAS1SMN1; SMN2LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4359475-A SPERMICIDES, MICROBIOCIDES OR ANTICONVULSANTS SYNTEX (U.S.A.) INC. (US) 1982-11-16 US disclosed
EP-0049565-A2 Derivatives of substituted N-alkylimidazoles, their preparation and pharmaceutical compositions containing them SYNTEX (U.S.A.) INC. (US) 1982-04-14 EP disclosed
US-4321272-A Derivatives of substituted N-alkylimidazoles SYNTEX (U.S.A.) INC. (US) 1982-03-23 US disclosed