SCHEMBL11255382

SCHEMBL11255382

CCCn1c(-c2ccc(NC(C)=O)cc2)cc2cc(O)ccc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 3/20 0.45
MEN1 O00255 4/20 0.44
ALDH1A1 P00352 4/20 0.44
KMT2A Q03164 4/20 0.44
MAPT P10636 4/20 0.44
CA12 O43570 1/20 0.44
BRD4 O60885 1/20 0.44
NR1I2 O75469 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
MB P02144 1/20 0.44
CYP1A1 P04798 1/20 0.44
CA3 P07451 1/20 0.44
CYP3A4 P08684 1/20 0.44
RARG P13631 1/20 0.44
TSHR P16473 1/20 0.44
ALOX5AP P20292 1/20 0.44
CA4 P22748 1/20 0.44
CA7 P43166 1/20 0.44
NR1I3 Q14994 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11258892 0.79 ALDH1A1 (0.51) ADORA2BMEN1ALDH1A1KMT2AESR1
SCHEMBL11259021 0.78 PPARA (0.42) ADORA2BMEN1ALDH1A1KMT2AMAPT
SCHEMBL11257361 0.73 MTNR1A (0.45) ADORA2BMEN1ALDH1A1KMT2AMAPT
SCHEMBL11257688 0.71 PPARA (0.42) ADORA2BMEN1ALDH1A1KMT2AMAPT
Acetaminophen SCHEMBL17114004 0.69 KMT2A (0.91) MEN1ALDH1A1KMT2AMAPTCA12
SCHEMBL16167713 0.68 MTNR1A (0.48) ADORA2BALDH1A1KMT2ANR1I2L3MBTL1
SCHEMBL2605857 0.68 KMT2A (0.87) MEN1ALDH1A1KMT2AMAPTCA12
SCHEMBL11251055 0.68 ESR1 (0.44) ADORA2BMEN1ALDH1A1KMT2AMAPT
SCHEMBL27761990 0.67 ALDH1A1 (0.51) MEN1ALDH1A1KMT2AESR1SMN1; SMN2
SCHEMBL1808467 0.67 MEN1 (0.64) MEN1ALDH1A1KMT2AMAPTCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0015523-B1 INDOLE DERIVATIVES, THEIR PREPARATION AND THEIR USE FOR MEDICAMENTS Dr. Karl Thomae GmbH (DE) 1982-10-13 EP disclosed
US-4343811-A ATHEROSCLEROSIS BOEHRINGER INGELHEIM GMBH (DE) 1982-08-10 US disclosed
EP-0015523-A1 Indole derivatives, their preparation and their use for medicaments Dr. Karl Thomae GmbH (DE) 1980-09-17 EP disclosed