SCHEMBL11255428

SCHEMBL11255428

CC1(C)CCc2cc(Cl)cc(-c3nc4ccncc4[nH]3)c2O1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 2/20 0.44
HPGD P15428 2/20 0.44
PKM P14618 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
PDE5A O76074 4/20 0.41
JMJD6 Q6NYC1 1/20 0.40
RPS6KA5 O75582 1/20 0.39
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
AURKA O14965 1/20 0.37
NR3C1 P04150 1/20 0.37
PGR P06401 1/20 0.37
NR3C2 P08235 1/20 0.37
METAP1 P53582 2/20 0.36
METAP2 P50579 1/20 0.36
HPSE Q9Y251 1/20 0.35
ADORA3 P0DMS8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11253114 0.86 AMY1A (0.47) ALDH1A1KDM4EHPGDPKMNPC1
SCHEMBL11262388 0.84 AMY1A (0.37) ALDH1A1KDM4EHPGDAMY1A
SCHEMBL11252873 0.84 PDE5A (0.48) ALDH1A1KDM4EHPGDPKMNPC1
SCHEMBL11262531 0.83 AMY1A (0.41) NPC1RAB9AAMY1A
SCHEMBL11259880 0.82 AMY1A (0.51) NPC1RAB9AMETAP1METAP2HPSE
SCHEMBL11266547 0.79 RHEB (0.31)
Hydrochloric Acid SCHEMBL11264419 0.78 PDE5A (0.43) ALDH1A1KDM4EHPGDPDE5APDE3B
SCHEMBL11261992 0.78 METAP2 (0.33) NPC1RAB9AMETAP1METAP2
SCHEMBL11264095 0.77 AMY1A (0.34) ALDH1A1KDM4ENPC1RAB9AAMY1A
SCHEMBL11256562 0.75 PDE5A (0.38) ALDH1A1KDM4EHPGDPKMNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4329459-A ENDOPEROXIDE CYCLOXGENASE INHIBITORS THE UPJOHN COMPANY (US) 1982-05-11 US claimed
US-4329459-A ENDOPEROXIDE CYCLOXGENASE INHIBITORS THE UPJOHN COMPANY (US) 1982-05-11 US disclosed