SCHEMBL11255431

SCHEMBL11255431

CC(C(=O)O)c1cccc2c(-c3ccc(Cl)cc3)nccc12

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SELPLG Q14242 1/20 0.44
CSNK2A2 P19784 2/20 0.43
CSNK2B P67870 2/20 0.43
IDO1 P14902 1/20 0.41
TDO2 P48775 1/20 0.41
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
CXCL8 P10145 1/20 0.39
LMNA P02545 1/20 0.37
TRPV1 Q8NER1 1/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2C8 P10632 1/20 0.36
CYP2C9 P11712 1/20 0.36
DHODH Q02127 1/20 0.36
MAOA P21397 1/20 0.36
ADRA1A P35348 1/20 0.36
KMO O15229 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11256929 0.88 RAB9A (0.40) LMNATRPV1CYP3A4DHODH
SCHEMBL11259590 0.87 TRPV1 (0.37) SELPLGCXCL8TRPV1CYP3A4CYP2C9
SCHEMBL11257836 0.87 BCHE (0.41) CSNK2A2CSNK2BPDE3BPDE3ADHODH
SCHEMBL11257378 0.85 MMP2 (0.48) PDE3BPDE3ALMNA
SCHEMBL11257643 0.85 PSEN1 (0.39) LMNACYP3A4CYP2C9
SCHEMBL11263420 0.85 HSP90AA1 (0.37) CXCL8TRPV1
SCHEMBL11439308 0.81 CXCL8 (0.46) CXCL8CYP3A4CYP2C9
SCHEMBL11254442 0.78 KDM4E (0.38)
SCHEMBL11260467 0.78 TDO2 (0.42) SELPLGCSNK2A2CSNK2BIDO1TDO2
SCHEMBL298816 0.76 CYP2A6 (0.40) TDO2CXCL8CYP3A4MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337256-A ANTIINFLAMMATORY AGENTS; ANTIAGGLOMERANTS; ENZYME INHIBITORS; ANTIULCER AGENTS TEIKOKU HORMONE MANUFACTURING CO., LTD. (JP) 1982-06-29 US disclosed
EP-0013411-A1 Isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-07-23 EP disclosed