SCHEMBL11255436

SCHEMBL11255436

Oc1ccc2c(c1)c(-c1ccncc1)c1n2CCCCC1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.50
ALDH1A1 P00352 2/20 0.50
ALOX15 P16050 1/20 0.50
ALOX5 P09917 2/20 0.44
PTGS1 P23219 1/20 0.44
PTGS2 P35354 1/20 0.44
MAPK1 P28482 1/20 0.44
THRB P10828 1/20 0.36
HTT P42858 1/20 0.36
ESR1 P03372 8/20 0.35
ESR2 Q92731 2/20 0.35
QPCT Q16769 1/20 0.34
MEN1 O00255 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
HTR6 P50406 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11260529 0.99 GAA (0.48) GAAALDH1A1ALOX15ALOX5PTGS1
SCHEMBL11500212 0.95 GAA (0.47) GAAALDH1A1ALOX15ALOX5PTGS1
SCHEMBL11262244 0.90 GAA (0.42) GAAALDH1A1ALOX15ALOX5PTGS1
SCHEMBL11250873 0.86 GAA (0.52) GAAALDH1A1ALOX15ALOX5PTGS1
SCHEMBL11263577 0.81 GAA (0.47) GAAALDH1A1ALOX15ALOX5PTGS1
SCHEMBL11260420 0.76 GAA (0.39) GAAALDH1A1ALOX15MAPK1MEN1
SCHEMBL11250723 0.75 GAA (0.44) GAAALDH1A1ALOX15ALOX5PTGS1
SCHEMBL11269896 0.75 GAA (0.38) GAAALDH1A1ALOX15MAPK1MEN1
SCHEMBL11269891 0.74 HTR6 (0.38) GAAALDH1A1ALOX15MAPK1MEN1
SCHEMBL11267995 0.74 ADORA3 (0.40) GAAALDH1A1ALOX15ALOX5THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0015523-B1 INDOLE DERIVATIVES, THEIR PREPARATION AND THEIR USE FOR MEDICAMENTS Dr. Karl Thomae GmbH (DE) 1982-10-13 EP disclosed
US-4343811-A ATHEROSCLEROSIS BOEHRINGER INGELHEIM GMBH (DE) 1982-08-10 US disclosed
EP-0015523-A1 Indole derivatives, their preparation and their use for medicaments Dr. Karl Thomae GmbH (DE) 1980-09-17 EP disclosed