SCHEMBL11263577

SCHEMBL11263577

Oc1ccc2c(c1)c(-c1ccccn1)c1n2CCCCC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.47
ALDH1A1 P00352 2/20 0.47
ALOX15 P16050 1/20 0.47
TGFBR1 P36897 6/20 0.45
MAPK1 P28482 2/20 0.41
ALOX5 P09917 1/20 0.41
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
METAP1 P53582 3/20 0.38
THRB P10828 2/20 0.37
TGFBR2 P37173 2/20 0.37
MAP3K20 Q9NYL2 2/20 0.37
CYP2C9 P11712 1/20 0.37
MAPK14 Q16539 1/20 0.35
CNR2 P34972 1/20 0.35
LMNA P02545 1/20 0.35
TSHR P16473 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11250723 0.81 GAA (0.44) GAAALDH1A1ALOX15MAPK1ALOX5
SCHEMBL11255436 0.81 GAA (0.50) GAAALDH1A1ALOX15MAPK1ALOX5
SCHEMBL11260529 0.80 GAA (0.48) GAAALDH1A1ALOX15MAPK1ALOX5
SCHEMBL11500212 0.77 GAA (0.47) GAAALDH1A1ALOX15MAPK1ALOX5
SCHEMBL11264505 0.69 GAA (0.41) GAAALDH1A1ALOX15CYP2C9LMNA
SCHEMBL21158689 0.67 HTR2A (0.39) TGFBR1THRBMAPK14KMT2AHTT
SCHEMBL12743756 0.64 TGFBR1 (0.35) GAAALDH1A1TGFBR1MAPK1KMT2A
SCHEMBL569668 0.64 ALOX5 (0.44) TGFBR1ALOX5THRBMAPK14
SCHEMBL23926385 0.63 ADORA3 (0.39) GAAALDH1A1TGFBR1MAPK1METAP1
SCHEMBL6068182 0.62 KDM1A (0.54) ALDH1A1ALOX15MAPK1ALOX5METAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0015523-B1 INDOLE DERIVATIVES, THEIR PREPARATION AND THEIR USE FOR MEDICAMENTS Dr. Karl Thomae GmbH (DE) 1982-10-13 EP disclosed
US-4343811-A ATHEROSCLEROSIS BOEHRINGER INGELHEIM GMBH (DE) 1982-08-10 US disclosed
EP-0015523-A1 Indole derivatives, their preparation and their use for medicaments Dr. Karl Thomae GmbH (DE) 1980-09-17 EP disclosed