SCHEMBL11259602

SCHEMBL11259602

CN(C(=N)NC(=O)NC(C)(C)C)c1ccc(Cl)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.42
HTT P42858 2/20 0.40
POLB P06746 2/20 0.40
MAPT P10636 1/20 0.39
ALDH1A1 P00352 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
KDM4E B2RXH2 1/20 0.38
HSD17B10 Q99714 1/20 0.38
LMNA P02545 1/20 0.36
MAPK1 P28482 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
LIPE Q05469 1/20 0.36
MAPK13 O15264 1/20 0.36
MAPK12 P53778 1/20 0.36
MAPK11 Q15759 1/20 0.36
MAPK14 Q16539 1/20 0.36
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11252555 0.89 TRPA1 (0.38) TRPA1HTTPOLBMAPTALDH1A1
SCHEMBL11055797 0.78 MAPK1 (0.48) HTTPOLBALDH1A1KDM4ELMNA
Hydrochloric Acid SCHEMBL11250652 0.77 POLB (0.41) POLBMAPTALDH1A1TDP1KDM4E
SCHEMBL11721893 0.75 HTT (0.38) TRPA1HTTPOLBALDH1A1KDM4E
SCHEMBL14868762 0.74 HTR3E (0.41) POLBMAPTALDH1A1TDP1KDM4E
SCHEMBL11255033 0.73 TSHR (0.42) POLBMAPTALDH1A1LMNAMAPK1
SCHEMBL11054637 0.73 HTT (0.52) TRPA1HTTMAPTALDH1A1TDP1
Hydrochloric Acid SCHEMBL11249260 0.72 HTT (0.38) HTTPOLBALDH1A1KDM4ELMNA
SCHEMBL11838675 0.72 ALDH1A1 (0.41) POLBMAPTALDH1A1TDP1KDM4E
SCHEMBL19891465 0.71 LMNA (0.42) TRPA1POLBMAPTALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4326074-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4025652-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1977-05-24 US disclosed