SCHEMBL11260065

SCHEMBL11260065

CCOC(=O)Cn1c(=O)n(Cc2ccc3ccccc3c2)c2ccccc21

nearest known ligand 0.69

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.69
TSHR P16473 1/20 0.54
KMT2A Q03164 6/20 0.53
MAPT P10636 2/20 0.53
MEN1 O00255 5/20 0.53
GAA P10253 2/20 0.53
LMNA P02545 2/20 0.53
HTT P42858 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
L3MBTL1 Q9Y468 2/20 0.52
TP53 P04637 1/20 0.52
KDM4E B2RXH2 2/20 0.50
RAB9A P51151 1/20 0.50
GLA P06280 1/20 0.50
NOD2 Q9HC29 1/20 0.47
NOD1 Q9Y239 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10487824 0.90 ALDH1A1 (0.58) ALDH1A1TSHRKMT2AMAPTMEN1
SCHEMBL11253338 0.85 ALDH1A1 (0.76) ALDH1A1TSHRKMT2AMAPTMEN1
SCHEMBL7734714 0.85 ALDH1A1 (0.81) ALDH1A1TSHRKMT2AMAPTMEN1
SCHEMBL11262526 0.85 LMNA (0.73) ALDH1A1TSHRKMT2AMAPTMEN1
SCHEMBL11263773 0.84 MEN1 (0.72) ALDH1A1TSHRKMT2AMAPTMEN1
SCHEMBL11258740 0.84 ALDH1A1 (0.74) ALDH1A1TSHRKMT2AMAPTMEN1
SCHEMBL11264725 0.82 APEX1 (0.64) KMT2AMEN1SMN1; SMN2L3MBTL1KDM4E
SCHEMBL1857784 0.81 VDR (0.50) ALDH1A1KMT2AMAPTMEN1GAA
SCHEMBL7740712 0.79 ALDH1A1 (0.66) ALDH1A1TSHRKMT2AMAPTMEN1
SCHEMBL11266490 0.79 ALDH1A1 (0.69) ALDH1A1TSHRKMT2AMEN1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0019440-B1 BENZIMIDAZOLONE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM PFIZER INC. (US) 1982-09-29 EP disclosed
EP-0019440-A1 Benzimidazolone derivatives, process for their preparation and pharmaceutical compositions containing them PFIZER INC. (US) 1980-11-26 EP disclosed
US-4209527-A ANTIDIABETIC AGENTS PFIZER INC. (US) 1980-06-24 US disclosed