SCHEMBL11261633

SCHEMBL11261633

Cc1cccc(C)c1NC(=S)NC(N)=O

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 4/20 0.58
ALDH1A1 P00352 3/20 0.58
ALOX12 P18054 2/20 0.56
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
DRD2 P14416 1/20 0.54
HTR2A P28223 1/20 0.54
HTR2B P41595 1/20 0.54
PKM P14618 1/20 0.53
GAA P10253 2/20 0.50
LMNA P02545 1/20 0.50
ATM Q13315 1/20 0.49
EPHX1 P07099 1/20 0.47
MAPT P10636 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11051530 0.82 GAA (0.50) POLBALDH1A1ALOX12CYP1A2CYP3A4
SCHEMBL5520683 0.81 DRD2 (0.59) POLBALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL5222474 0.81 GRIN2D (0.55) POLBALDH1A1ALOX12CYP1A2DRD2
SCHEMBL15484311 0.80 LMNA (0.69) POLBALDH1A1ALOX12CYP1A2CYP3A4
SCHEMBL6692615 0.79 DRD2 (0.54) POLBALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL11054164 0.79 GAA (0.50) CYP1A2GAA
SCHEMBL27709153 0.78 POLB (0.55) POLBALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL11258013 0.78 EPHX1 (0.72) ALDH1A1ALOX12CYP1A2CYP3A4CYP2C9
SCHEMBL8721848 0.78 POLB (0.53) POLBALDH1A1ALOX12CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL11258555 0.77 PKM (0.55) POLBALDH1A1CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4326074-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4115564-A Treatment of diarrhea with amidinoureas WILLIAM H. RORER, INC. (US) 1978-09-19 US disclosed
US-4025652-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1977-05-24 US disclosed