SCHEMBL11249519

SCHEMBL11249519

OCc1cccc2c(-c3ccc(Br)cc3)nccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 3/20 0.41
LMNA P02545 2/20 0.41
MAPT P10636 2/20 0.41
TP53 P04637 1/20 0.41
TSHR P16473 1/20 0.41
ALOX12 P18054 1/20 0.41
IDO1 P14902 3/20 0.36
TDO2 P48775 3/20 0.36
ALDH1A1 P00352 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
PDE5A O76074 1/20 0.35
ROS1 P08922 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11258335 0.88 ALDH1A1 (0.39) NPC1RAB9AMEN1KMT2AKDM4E
SCHEMBL11256693 0.88 ALDH1A1 (0.39) NPC1RAB9AMEN1KMT2AKDM4E
SCHEMBL11257847 0.85 HTR2B (0.45) NPC1RAB9AKMT2AKDM4ELMNA
SCHEMBL11254310 0.84 MEN1 (0.43) NPC1RAB9AMEN1KMT2AKDM4E
SCHEMBL11261678 0.84 TDP1 (0.45) NPC1RAB9AMEN1KMT2AKDM4E
SCHEMBL11261674 0.82 TDO2 (0.36) NPC1RAB9AMEN1KMT2AIDO1
SCHEMBL11253776 0.80 ROS1 (0.41) RAB9AMEN1KMT2AKDM4ELMNA
SCHEMBL11257966 0.80 ROS1 (0.46) MEN1KMT2AKDM4EMAPTALDH1A1
SCHEMBL11266092 0.80 ROS1 (0.37) MAPTALDH1A1ROS1RPS6KB1GAA
SCHEMBL11500393 0.79 PTGDR2 (0.45) MEN1KMT2AKDM4ELMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337256-A ANTIINFLAMMATORY AGENTS; ANTIAGGLOMERANTS; ENZYME INHIBITORS; ANTIULCER AGENTS TEIKOKU HORMONE MANUFACTURING CO., LTD. (JP) 1982-06-29 US disclosed
EP-0013411-A1 Isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-07-23 EP disclosed