SCHEMBL11265101

SCHEMBL11265101

COC(=S)c1cc(C)ccc1N

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 3/20 0.45
CYP3A4 P08684 2/20 0.45
TDP1 Q9NUW8 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
TP53 P04637 1/20 0.45
THRB P10828 1/20 0.45
MAPT P10636 4/20 0.44
HTT P42858 2/20 0.44
NPC1 O15118 2/20 0.44
MAPK1 P28482 1/20 0.44
ALDH1A1 P00352 7/20 0.42
HSD17B10 Q99714 3/20 0.41
GAA P10253 3/20 0.39
KDM4E B2RXH2 2/20 0.39
HPGD P15428 2/20 0.39
TSHR P16473 2/20 0.39
CYP1A2 P05177 1/20 0.38
CFTR P13569 1/20 0.36
CA1 P00915 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11263870 0.98 ALOX15 (0.43) ALOX15CYP3A4TDP1SMN1; SMN2TP53
SCHEMBL11714480 0.79 ABL1 (0.50) ALOX15CYP3A4TDP1SMN1; SMN2MAPT
SCHEMBL10373446 0.78 CSNK2A1 (0.52) ALOX15TDP1SMN1; SMN2TP53MAPT
SCHEMBL7001137 0.78 ACHE (0.54) CYP3A4SMN1; SMN2MAPTALDH1A1HSD17B10
SCHEMBL9770532 0.78 ALOX15 (0.50) ALOX15CYP3A4TDP1SMN1; SMN2TP53
SCHEMBL8071051 0.78 TDP1 (0.50) ALOX15CYP3A4TDP1SMN1; SMN2TP53
SCHEMBL1129416 0.77 ALDH1A1 (0.64) ALOX15CYP3A4TDP1SMN1; SMN2TP53
SCHEMBL11162396 0.77 ALOX15 (0.45) ALOX15CYP3A4TDP1SMN1; SMN2TP53
SCHEMBL27721513 0.77 CPS1 (0.38) SMN1; SMN2MAPTNPC1ALDH1A1GAA
SCHEMBL4098055 0.74 IDO1 (0.47) TDP1SMN1; SMN2TP53MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4348396-A Substituted 11-oxo-11H-pyrido[2,1-b]quinazolines and method of inhibiting allergic reactions with them HOFFMANN-LA ROCHE INC. (US) 1982-09-07 US disclosed
US-4282360-A ANTIALLERGENS HOFFMANN-LA ROCHE INC. (US) 1981-08-04 US disclosed
EP-0027268-A2 Quinazoline derivatives, process and intermediates for their preparation, medicaments containing them and their pharmaceutical use F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1981-04-22 EP disclosed