SCHEMBL11265463

SCHEMBL11265463

O=C(c1ccccc1)c1ccccc1NCC(O)CCl

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.57
PPARG P37231 3/20 0.49
KMT2A Q03164 1/20 0.48
BACE1 P56817 1/20 0.47
KDM4E B2RXH2 1/20 0.45
AGTR1 P30556 1/20 0.45
RAB9A P51151 1/20 0.45
AKR1C3 P42330 1/20 0.43
TLR4 O00206 1/20 0.43
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 2/20 0.40
HSD17B10 Q99714 2/20 0.40
POLB P06746 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
ABCB1 P08183 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11275701 0.87 ALDH1A1 (0.49) ALDH1A1PPARGKMT2ABACE1KDM4E
SCHEMBL14746862 0.86 ALDH1A1 (0.54) ALDH1A1PPARGKMT2ABACE1KDM4E
SCHEMBL11272884 0.85 PPARG (0.67) ALDH1A1PPARGKMT2AKDM4ETLR4
SCHEMBL14982070 0.79 ALDH1A1 (0.51) ALDH1A1PPARGKMT2AKDM4EAGTR1
SCHEMBL10735844 0.79 LMNA (0.49) ALDH1A1KMT2AKDM4ERAB9AGAA
SCHEMBL27388643 0.79 KMT2A (0.51) ALDH1A1PPARGKMT2AKDM4EAGTR1
SCHEMBL10954896 0.79 KDM4E (0.59) ALDH1A1KMT2AKDM4EGAAMAPT
SCHEMBL1532856 0.76 KMT2A (0.58) ALDH1A1KMT2AKDM4EAGTR1RAB9A
SCHEMBL698881 0.76 AGTR1 (0.60) ALDH1A1PPARGKMT2AKDM4EAGTR1
SCHEMBL6274259 0.75 ALDH1A1 (0.46) ALDH1A1PPARGKMT2ABACE1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0004024-B1 METHOD FOR PREPARING 3-HYDROXY-6-PHENYL-1,2,3,4-TETRAHYDRO-1,5-BENZODIAZOCINES Kali-Chemie Pharma GmbH (DE) 1982-02-24 EP disclosed
EP-0004024-A2 Method for preparing 3-hydroxy-6-phenyl-1,2,3,4-tetrahydro-1,5-benzodiazocines Kali-Chemie Pharma GmbH (DE) 1979-09-19 EP disclosed