SCHEMBL11265709

SCHEMBL11265709

COc1nc2cc(-c3ccncc3)ccc2[nH]1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 3/20 0.45
PDE3A Q14432 3/20 0.45
CLK1 P49759 2/20 0.44
GAK O14976 1/20 0.43
TLR9 Q9NR96 1/20 0.42
TLR8 Q9NR97 1/20 0.42
TLR7 Q9NYK1 1/20 0.42
MMP2 P08253 1/20 0.42
MMP13 P45452 1/20 0.42
MMP14 P50281 1/20 0.42
AAK1 Q2M2I8 4/20 0.42
PDGFRB P09619 3/20 0.40
PDGFRA P16234 3/20 0.40
JAK2 O60674 1/20 0.40
RAF1 P04049 2/20 0.39
MAPK13 O15264 1/20 0.39
MAPK12 P53778 1/20 0.39
MAPK11 Q15759 1/20 0.39
MAPK14 Q16539 1/20 0.39
DYRK1A Q13627 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11271918 0.85 MMP2 (0.49) PDE3BPDE3ACLK1TLR9TLR8
Water SCHEMBL11275606 0.84 MMP2 (0.48) PDE3BPDE3ACLK1TLR9TLR8
SCHEMBL11269561 0.81 CYP3A4 (0.44) PDE3BPDE3ACLK1TLR9TLR8
SCHEMBL11273096 0.80 CYP2D6 (0.54) PDE3BPDE3ACLK1TLR9TLR8
SCHEMBL11221691 0.79 PDE3B (0.49) PDE3BPDE3ACLK1MMP2MMP13
SCHEMBL11270335 0.78 CYP3A4 (0.48) PDE3BPDE3ACLK1TLR9TLR8
SCHEMBL31265084 0.76 MMP2 (0.49) PDE3BPDE3ACLK1MMP2MMP13
SCHEMBL17493786 0.76 PDE3B (0.49) PDE3BPDE3ACLK1MMP2MMP13
SCHEMBL16848371 0.76 JAK2 (0.50) PDE3BPDE3ACLK1AAK1JAK2
SCHEMBL11269149 0.76 PDE3B (0.49) PDE3BPDE3ACLK1MMP2MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0055453-A2 5-(Pyridinyl)-benzimidazole derivatives and preparation STERLING DRUG INC. (US) 1982-07-07 EP disclosed
US-4335132-A 5-(Py-Y)-1H-benzimidazol-2-ols and 5-(Py-Y-)-1H-benzimidazole-2-thiols STERLING DRUG, INC. (US) 1982-06-15 US disclosed