SCHEMBL11269561

SCHEMBL11269561

CCCOc1nc2cc(-c3ccncc3)ccc2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
MMP2 P08253 1/20 0.43
MMP13 P45452 1/20 0.43
MMP14 P50281 1/20 0.43
PDE3B Q13370 2/20 0.43
PDE3A Q14432 2/20 0.43
KDM4E B2RXH2 1/20 0.41
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HSD17B10 Q99714 1/20 0.41
S1PR1 P21453 1/20 0.40
S1PR3 Q99500 1/20 0.40
GCGR P47871 4/20 0.40
MAPK14 Q16539 2/20 0.40
MAPK13 O15264 1/20 0.40
MAPK12 P53778 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11273096 0.93 CYP2D6 (0.54) CYP3A4CYP2D6MMP2MMP13MMP14
SCHEMBL11270335 0.91 CYP3A4 (0.48) CYP3A4CYP2D6MMP2MMP13MMP14
SCHEMBL11271918 0.90 MMP2 (0.49) CYP3A4CYP2D6MMP2MMP13MMP14
Water SCHEMBL11275606 0.89 MMP2 (0.48) CYP3A4CYP2D6MMP2MMP13MMP14
SCHEMBL11265709 0.81 PDE3B (0.45) CYP3A4CYP2D6MMP2MMP13MMP14
SCHEMBL11275736 0.77 ABL1 (0.45) MMP2MMP13MMP14GCGRMAPK14
SCHEMBL11218846 0.76 AAK1 (0.53) CYP3A4CYP2D6MMP2MMP13MMP14
SCHEMBL11270413 0.75 CYP11B2 (0.58) CYP3A4CYP2D6MMP2MMP13MMP14
SCHEMBL11271873 0.73 KDM4C (0.39) MMP2MMP13MMP14PDE3BPDE3A
SCHEMBL3974150 0.73 RAB9A (0.53) CYP2D6KDM4ENPC1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0055453-A2 5-(Pyridinyl)-benzimidazole derivatives and preparation STERLING DRUG INC. (US) 1982-07-07 EP disclosed
US-4335132-A 5-(Py-Y)-1H-benzimidazol-2-ols and 5-(Py-Y-)-1H-benzimidazole-2-thiols STERLING DRUG, INC. (US) 1982-06-15 US disclosed