SCHEMBL11273096

SCHEMBL11273096

CCCCOc1nc2cc(-c3ccncc3)ccc2[nH]1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.54
CYP3A4 P08684 2/20 0.54
GSK3B P49841 2/20 0.44
CDC7 O00311 1/20 0.44
ROCK2 O75116 1/20 0.44
MAP4K4 O95819 1/20 0.44
PIM1 P11309 1/20 0.44
PRKACA P17612 1/20 0.44
CDK2 P24941 1/20 0.44
HIPK2 Q9H2X6 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
IRAK4 Q9NWZ3 1/20 0.44
KDM4E B2RXH2 1/20 0.43
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
TSHR P16473 1/20 0.43
RAB9A P51151 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11270335 0.95 CYP3A4 (0.48) CYP2D6CYP3A4GSK3BCDC7ROCK2
SCHEMBL11269561 0.93 CYP3A4 (0.44) CYP2D6CYP3A4GSK3BCDC7ROCK2
SCHEMBL11271918 0.89 MMP2 (0.49) CYP2D6CYP3A4KDM4ENPC1ALDH1A1
Water SCHEMBL11275606 0.88 MMP2 (0.48) CYP2D6CYP3A4KDM4ENPC1ALDH1A1
SCHEMBL11265709 0.80 PDE3B (0.45) CYP2D6CYP3A4KDM4EALDH1A1HSD17B10
SCHEMBL11275736 0.76 ABL1 (0.45) MAP4K4MMP2MMP13MMP14GCGR
SCHEMBL11218846 0.75 AAK1 (0.53) CYP2D6CYP3A4KDM4EALDH1A1HSD17B10
SCHEMBL11270413 0.74 CYP11B2 (0.58) CYP2D6CYP3A4KDM4ENPC1ALDH1A1
SCHEMBL11271873 0.72 KDM4C (0.39) KDM4ENPC1ALDH1A1LMNAMAPT
SCHEMBL11221691 0.72 PDE3B (0.49) CYP2D6CYP3A4GSK3BCDC7KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0055453-A2 5-(Pyridinyl)-benzimidazole derivatives and preparation STERLING DRUG INC. (US) 1982-07-07 EP disclosed
US-4335132-A 5-(Py-Y)-1H-benzimidazol-2-ols and 5-(Py-Y-)-1H-benzimidazole-2-thiols STERLING DRUG, INC. (US) 1982-06-15 US disclosed