SCHEMBL1126602

SCHEMBL1126602

CCc1ccnc(N2CCN(c3ccc(NC(=O)C(=O)c4c(-c5cccs5)c(C)cn4C)cc3)CC2)c1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
DRD3 P35462 1/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
REV1 Q9UBZ9 3/20 0.37
MAPT P10636 6/20 0.37
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 3/20 0.37
POLB P06746 2/20 0.37
CYP2C19 P33261 1/20 0.37
KMT2A Q03164 3/20 0.36
HTT P42858 1/20 0.36
TP53 P04637 1/20 0.35
THRB P10828 1/20 0.35
FLT3 P36888 1/20 0.35
MEN1 O00255 2/20 0.34
MCHR1 Q99705 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1993070 0.85 MAPT (0.39) DRD2DRD4DRD3NPC1RAB9A
SCHEMBL1992803 0.76 REV1 (0.44) DRD2DRD4DRD3NPC1RAB9A
SCHEMBL1991665 0.75 HCRTR1 (0.44) DRD2DRD4DRD3NPC1RAB9A
SCHEMBL1996541 0.73 REV1 (0.40) DRD2DRD4DRD3SMN1; SMN2REV1
SCHEMBL1997118 0.73 ALDH1A1 (0.46) DRD2DRD4DRD3NPC1RAB9A
SCHEMBL1646298 0.71 THRB (0.51) DRD2DRD4DRD3SMN1; SMN2REV1
SCHEMBL1646885 0.71 DRD2 (0.43) DRD2DRD4DRD3SMN1; SMN2REV1
SCHEMBL1995053 0.70 MAPT (0.40) NPC1RAB9ASMN1; SMN2MAPTALDH1A1
SCHEMBL1991453 0.70 REV1 (0.42) DRD2DRD4DRD3NPC1RAB9A
SCHEMBL1645652 0.70 REV1 (0.43) DRD2DRD4DRD3SMN1; SMN2REV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2283006-A1 PYRROLE ANTIFUNGAL AGENTS F2G Limited (GB) 2011-02-16 EP disclosed
WO-2009130481-A1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2009-10-29 WO disclosed