SCHEMBL11267176

SCHEMBL11267176

O=c1n(CCCN2CC=C(c3ccc(Cl)cc3)CC2)nc2ccccn12

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.57
SIGMAR1 Q99720 6/20 0.57
DRD2 P14416 5/20 0.57
HTR2A P28223 5/20 0.57
KDM4E B2RXH2 2/20 0.57
ALDH1A1 P00352 2/20 0.57
HPGD P15428 2/20 0.57
HSD17B10 Q99714 2/20 0.57
ABCB11 O95342 1/20 0.57
LMNA P02545 1/20 0.57
ADRA2A P08913 1/20 0.57
CYP2D6 P10635 1/20 0.57
ADRA2B P18089 1/20 0.57
ADRA2C P18825 1/20 0.57
DRD1 P21728 1/20 0.57
DRD4 P21917 1/20 0.57
HRH2 P25021 1/20 0.57
ADRA1D P25100 1/20 0.57
TACR1 P25103 1/20 0.57
HTR2C P28335 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11267488 0.91 HTR1A (0.51) HTR1ASIGMAR1DRD2HTR2AKDM4E
SCHEMBL11264673 0.83 KDM4E (0.51) HTR1ASIGMAR1DRD2HTR2AKDM4E
SCHEMBL4865321 0.79 DRD2 (0.59) HTR1ASIGMAR1DRD2HTR2AKDM4E
SCHEMBL30767207 0.79 HTR1A (0.80) HTR1ASIGMAR1DRD2HTR2AKDM4E
Hydrochloric Acid SCHEMBL30945326 0.78 KDM4E (0.81) HTR1ASIGMAR1DRD2HTR2AKDM4E
SCHEMBL11262256 0.77 DRD2 (0.62) HTR1ASIGMAR1DRD2HTR2AKDM4E
SCHEMBL4868327 0.77 DRD2 (0.62) HTR1ASIGMAR1DRD2HTR2AKDM4E
SCHEMBL5846298 0.76 SIGMAR1 (0.68) HTR1ASIGMAR1DRD2HTR7PARP1
Hydrochloric Acid SCHEMBL5846785 0.75 SIGMAR1 (0.67) HTR1ASIGMAR1DRD2HTR7PARP1
SCHEMBL30764775 0.73 HTR1A (0.82) HTR1ASIGMAR1DRD2HTR2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4340597-A 1-Substituted-4-aryl-1,2,5,6-tetrahydro and hexahydropyridines SCHERING CORPORATION (US) 1982-07-20 US claimed
US-4340597-A 1-Substituted-4-aryl-1,2,5,6-tetrahydro and hexahydropyridines SCHERING CORPORATION (US) 1982-07-20 US disclosed