SCHEMBL11267643

SCHEMBL11267643

Clc1cccc2c1CCN=C2c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK10 P53779 8/20 0.49
CYP2A6 P11509 1/20 0.47
BCHE P06276 1/20 0.42
PTGS2 P35354 2/20 0.40
NR1I2 O75469 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
HTR2C P28335 1/20 0.40
ADRA1A P35348 1/20 0.40
OPRK1 P41145 1/20 0.40
CHRNA4 P43681 1/20 0.40
SLC6A3 Q01959 1/20 0.40
PDE4D Q08499 1/20 0.40
MAPK14 Q16539 2/20 0.40
MAPK9 P45984 1/20 0.40
PTGS1 P23219 1/20 0.39
HTR1A P08908 2/20 0.38
HTR7 P34969 2/20 0.38
HSD11B1 P28845 1/20 0.38
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11259543 0.86 MAPK10 (0.42) MAPK10MAPK14MAPK9HTR1AHTR7
SCHEMBL163051 0.77 MAPK10 (0.55) MAPK10CYP2A6MAPK14MAPK9
SCHEMBL29384557 0.77 MAPK10 (0.55) MAPK10CYP2A6MAPK14MAPK9
Hydrochloric Acid SCHEMBL27495714 0.75 MAPK10 (0.54) MAPK10MAPK14MAPK9
SCHEMBL29010816 0.74 MAPK10 (0.38) MAPK10BCHEADRA1AOPRK1PDE4D
SCHEMBL30167242 0.74 CYP19A1 (0.41) MAPK10BCHEHTR2CADRA1AMAPK14
SCHEMBL1010129 0.74 CYP19A1 (0.41) MAPK10BCHEHTR2CADRA1AMAPK14
SCHEMBL11261829 0.73 BRD4 (0.45) MAPK10PTGS2NR1I2ADORA3HTR2C
SCHEMBL14246803 0.73 ALDH1A1 (0.40) BCHEHTR1AHTR7NPC1RAB9A
SCHEMBL8215360 0.72 MAPK10 (0.62) MAPK10PTGS2NR1I2ADORA3HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337256-A ANTIINFLAMMATORY AGENTS; ANTIAGGLOMERANTS; ENZYME INHIBITORS; ANTIULCER AGENTS TEIKOKU HORMONE MANUFACTURING CO., LTD. (JP) 1982-06-29 US disclosed
EP-0013411-A1 Isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-07-23 EP disclosed