SCHEMBL1126895

SCHEMBL1126895

CC(Cc1cc(-c2ccccc2)c(C(=O)C(=O)Cl)[nH]1)Oc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39
PPARA Q07869 10/20 0.36
PPARG P37231 9/20 0.36
PRKAB2 O43741 3/20 0.35
PRKAG1 P54619 3/20 0.35
PRKAA2 P54646 3/20 0.35
PRKAA1 Q13131 3/20 0.35
PRKAG3 Q9UGI9 3/20 0.35
PRKAG2 Q9UGJ0 3/20 0.35
PRKAB1 Q9Y478 3/20 0.35
CYP1A2 P05177 1/20 0.35
GAA P10253 1/20 0.35
CYP2C9 P11712 1/20 0.35
PKM P14618 1/20 0.35
CYP2C19 P33261 1/20 0.35
MAPT P10636 1/20 0.35
CD274 Q9NZQ7 1/20 0.34
PTGER2 P43116 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1127401 0.81 CD274 (0.33) CYP1A2GAACYP2C9CYP2C19MAPT
SCHEMBL1127126 0.65 MTNR1A (0.41) MTNR1AMTNR1BPPARAPPARGCYP1A2
SCHEMBL17892031 0.62 MTNR1A (0.55) MTNR1AMTNR1BPRKAB2PRKAG1PRKAA2
SCHEMBL120055 0.62 MTNR1A (0.55) MTNR1AMTNR1BPRKAB2PRKAG1PRKAA2
SCHEMBL7566883 0.62 MTNR1A (0.55) MTNR1AMTNR1BPRKAB2PRKAG1PRKAA2
SCHEMBL28735087 0.62 SIGMAR1 (0.52) MTNR1AMTNR1BPPARAPPARG
SCHEMBL1418060 0.61 MTNR1A (0.59) MTNR1AMTNR1BCYP1A2GAACYP2C9
Acetic Acid SCHEMBL27633889 0.60 MTNR1A (0.62) MTNR1AMTNR1BCYP1A2GAACYP2C9
SCHEMBL7976612 0.60 CYP1A2 (0.58) MTNR1AMTNR1BPPARAPPARGPRKAB2
SCHEMBL11752459 0.60 CYP1A2 (0.58) MTNR1AMTNR1BPPARAPPARGPRKAB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2283006-A1 PYRROLE ANTIFUNGAL AGENTS F2G Limited (GB) 2011-02-16 EP disclosed
WO-2009130481-A1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2009-10-29 WO disclosed