SCHEMBL11269770

SCHEMBL11269770

CC(C)(C)NC(=O)NC(=N)Nc1cc(OCc2ccccc2)c(OCc2ccccc2)c(OCc2ccccc2)c1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.43
HPGD P15428 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
PPIA P62937 2/20 0.41
BRD4 O60885 1/20 0.41
SGMS2 Q8NHU3 1/20 0.40
LMNA P02545 1/20 0.40
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
RAB9A P51151 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
C5AR1 P21730 1/20 0.39
CTSV O60911 1/20 0.39
CTSL P07711 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11245263 0.89 C5AR1 (0.52) CYP19A1HPGDKDM4EALDH1A1PPIA
SCHEMBL11254295 0.82 SGMS2 (0.47) CYP19A1KDM4EPPIABRD4SGMS2
SCHEMBL11265930 0.81 C5AR1 (0.43) CYP19A1HPGDALDH1A1BRD4SGMS2
SCHEMBL11254409 0.81 GAA (0.41) HPGDKDM4EALDH1A1LMNANPC1
SCHEMBL11258028 0.81 C5AR1 (0.41) CYP19A1HPGDPPIABRD4SGMS2
SCHEMBL11280329 0.80 C5AR1 (0.47) KDM4ESGMS2C5AR1
SCHEMBL11284130 0.79 CYP19A1 (0.44) CYP19A1HPGDBRD4SGMS2LMNA
SCHEMBL7167350 0.78 PPIA (0.47) KDM4EPPIABRD4SGMS2C5AR1
SCHEMBL11275038 0.76 C5AR1 (0.47) MEN1KMT2AC5AR1
SCHEMBL11275041 0.76 C5AR1 (0.47) MEN1KMT2AC5AR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4326074-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed