SCHEMBL11280329

SCHEMBL11280329

N=C(N)NC(=N)Nc1cc(OCc2ccccc2)c(OCc2ccccc2)c(OCc2ccccc2)c1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
C5AR1 P21730 9/20 0.47
F10 P00742 2/20 0.41
MRGPRX1 Q96LB2 2/20 0.41
F9 P00740 1/20 0.41
F2 P00734 1/20 0.41
PRSS1 P07477 1/20 0.41
F7 P08709 1/20 0.41
SGMS2 Q8NHU3 1/20 0.40
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11254295 0.90 SGMS2 (0.47) C5AR1F10F2PRSS1F7
SCHEMBL11246834 0.89 C5AR1 (0.51) C5AR1F10MRGPRX1F9F2
SCHEMBL11138186 0.87 ALDH1A1 (0.48) C5AR1KDM4E
SCHEMBL7167350 0.87 PPIA (0.47) C5AR1SGMS2KDM4E
SCHEMBL11265836 0.87 C5AR1 (0.63) C5AR1F10MRGPRX1F2PRSS1
SCHEMBL11265930 0.86 C5AR1 (0.43) C5AR1SGMS2
SCHEMBL11284130 0.84 CYP19A1 (0.44) C5AR1SGMS2
SCHEMBL11275041 0.81 C5AR1 (0.47) C5AR1
SCHEMBL11275038 0.81 C5AR1 (0.47) C5AR1
SCHEMBL11269770 0.80 CYP19A1 (0.43) C5AR1SGMS2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4326075-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4203920-A ANTIDIARRHEAL WILLIAM H. RORER, INC. (US) 1980-05-20 US disclosed
US-4060635-A Amidinoureas for treating diarrhea WILLIAM H. RORER, INC. (US) 1977-11-29 US disclosed