SCHEMBL1127003

SCHEMBL1127003

O=C(O)CCc1c(-c2ccccc2)c[nH]c1C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GPR17 Q13304 10/20 0.54
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
FBP1 P09467 2/20 0.49
FFAR1 O14842 1/20 0.45
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
HSD17B10 Q99714 1/20 0.43
KEAP1 Q14145 1/20 0.42
PTGER1 P34995 1/20 0.41
PTGER4 P35408 1/20 0.41
PTGER3 P43115 1/20 0.41
PTGER2 P43116 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1126776 0.73 ALDH1A1 (0.53) KDM4EALDH1A1CYP1A2CYP2C9HSD17B10
SCHEMBL11172051 0.72 MAPT (0.49)
SCHEMBL14739748 0.71 GPR17 (1.00) GPR17KDM4EALDH1A1FBP1
SCHEMBL14739170 0.70 GPR17 (1.00) GPR17KDM4EALDH1A1FBP1
SCHEMBL2994014 0.69 PTGER4 (0.64) GPR17FFAR1CYP1A2CYP2C9HSD17B10
SCHEMBL11007304 0.68 PTGER1 (0.54) GPR17ALDH1A1FFAR1HSD17B10KEAP1
SCHEMBL8923388 0.68 KDM4E (0.43) KDM4EALDH1A1CYP1A2HSD17B10
SCHEMBL11162121 0.68 HTT (0.53) KDM4EALDH1A1CYP1A2
SCHEMBL31212507 0.67 PTGER4 (0.77) FFAR1KEAP1PTGER1PTGER4PTGER3
SCHEMBL1261128 0.67 PTGER4 (0.77) FFAR1KEAP1PTGER1PTGER4PTGER3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2283006-A1 PYRROLE ANTIFUNGAL AGENTS F2G Limited (GB) 2011-02-16 EP disclosed
WO-2009130481-A1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2009-10-29 WO disclosed