SCHEMBL1127235

SCHEMBL1127235

CCCOCCn1c(C)cc(-c2ccccc2)c1C(=O)C(=O)Cl

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.37
KDM4E B2RXH2 5/20 0.37
ALDH1A1 P00352 4/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
TDP1 Q9NUW8 1/20 0.37
TSHR P16473 2/20 0.35
SMN1; SMN2 Q16637 3/20 0.34
GAA P10253 2/20 0.34
LMNA P02545 1/20 0.34
HPGD P15428 1/20 0.34
NOTUM Q6P988 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
JMJD6 Q6NYC1 1/20 0.33
AR P10275 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1126938 0.92 KDM4E (0.43) THRBKDM4EALDH1A1MEN1KMT2A
SCHEMBL15161873 0.91 THRB (0.37) THRBKDM4EALDH1A1TSHRSMN1; SMN2
SCHEMBL1127378 0.86 HPGD (0.41) ALDH1A1TDP1TSHRSMN1; SMN2GAA
SCHEMBL1127595 0.86 KDM4E (0.39) KDM4EALDH1A1MEN1KMT2ATSHR
SCHEMBL15161860 0.85 LMNA (0.44) KDM4EALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL1127195 0.84 RARB (0.39) KDM4ETSHRGAAAR
SCHEMBL23488097 0.83 THRB (0.40) THRBKDM4EALDH1A1MEN1KMT2A
SCHEMBL1126982 0.83 TP53 (0.35) THRBKDM4EALDH1A1MEN1KMT2A
SCHEMBL1126775 0.83 ALDH1A1 (0.40) KDM4EALDH1A1KMT2ATDP1GAA
SCHEMBL1127423 0.83 TSHR (0.39) THRBKDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2283006-B1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2015-02-25 EP disclosed
EP-2626361-B1 Pyrrole antifungal agents F2G LTD (GB) 2014-10-15 EP disclosed
EP-2626361-A1 Pyrrole antifungal agents F2G Limited (GB) 2013-08-14 EP disclosed
EP-2283006-A1 PYRROLE ANTIFUNGAL AGENTS F2G Limited (GB) 2011-02-16 EP disclosed
WO-2009130481-A1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2009-10-29 WO disclosed