SCHEMBL1126938

SCHEMBL1126938

CCOCCn1c(C)cc(-c2ccccc2)c1C(=O)C(=O)Cl

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.43
TSHR P16473 3/20 0.38
ALDH1A1 P00352 4/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
GAA P10253 2/20 0.37
LMNA P02545 1/20 0.37
HPGD P15428 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
JMJD6 Q6NYC1 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
THRB P10828 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
GABRA2 P47869 1/20 0.35
GABRB2 P47870 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1127595 0.94 KDM4E (0.39) KDM4ETSHRALDH1A1SMN1; SMN2GAA
SCHEMBL1127235 0.92 THRB (0.37) KDM4ETSHRALDH1A1SMN1; SMN2GAA
SCHEMBL1127423 0.89 TSHR (0.39) KDM4ETSHRALDH1A1SMN1; SMN2GAA
SCHEMBL1127378 0.88 HPGD (0.41) TSHRALDH1A1SMN1; SMN2GAALMNA
SCHEMBL15161860 0.86 LMNA (0.44) KDM4EALDH1A1SMN1; SMN2LMNAHPGD
SCHEMBL23488097 0.84 THRB (0.40) KDM4ETSHRALDH1A1SMN1; SMN2GAA
SCHEMBL1126775 0.84 ALDH1A1 (0.40) KDM4EALDH1A1GAAHPGDKMT2A
SCHEMBL1126982 0.84 TP53 (0.35) KDM4ETSHRALDH1A1SMN1; SMN2GAA
SCHEMBL15161873 0.84 THRB (0.37) KDM4ETSHRALDH1A1SMN1; SMN2GAA
SCHEMBL1127780 0.83 KDM4E (0.39) KDM4EALDH1A1GAAHPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2283006-B1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2015-02-25 EP disclosed
EP-2626361-B1 Pyrrole antifungal agents F2G LTD (GB) 2014-10-15 EP disclosed
EP-2626361-A1 Pyrrole antifungal agents F2G Limited (GB) 2013-08-14 EP disclosed
EP-2283006-A1 PYRROLE ANTIFUNGAL AGENTS F2G Limited (GB) 2011-02-16 EP disclosed
WO-2009130481-A1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2009-10-29 WO disclosed