SCHEMBL1127247

SCHEMBL1127247

COCCc1c(-c2ccccc2)c[nH]c1C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.48
ADRB2 P07550 1/20 0.38
KDM4E B2RXH2 4/20 0.35
DYRK1A Q13627 2/20 0.35
CDC7 O00311 1/20 0.35
PLK4 O00444 1/20 0.35
CHEK1 O14757 1/20 0.35
CHUK O15111 1/20 0.35
PDPK1 O15530 1/20 0.35
DYRK3 O43781 1/20 0.35
ROCK2 O75116 1/20 0.35
PRKD3 O94806 1/20 0.35
MAP4K4 O95819 1/20 0.35
PAK4 O96013 1/20 0.35
NTRK1 P04629 1/20 0.35
PRKCG P05129 1/20 0.35
INSR P06213 1/20 0.35
LCK P06239 1/20 0.35
FYN P06241 1/20 0.35
CDK1 P06493 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1127088 0.92 HTT (0.47) HTTADRB2KDM4EDYRK1ACDC7
SCHEMBL1127206 0.91 HTT (0.46) HTTADRB2KDM4EDYRK1ACDC7
SCHEMBL1126842 0.84 HTT (0.42) HTTKDM4EDYRK1ACDC7PLK4
SCHEMBL1126705 0.83 HTT (0.50) HTTADRB2KDM4EDYRK1ACDC7
SCHEMBL1127356 0.83 HTT (0.41) HTTADRB2DYRK1ACDC7PLK4
SCHEMBL1127180 0.79 ADRB2 (0.40) HTTADRB2KDM4EDYRK1ACDC7
SCHEMBL1127151 0.76 HTT (0.43) HTTDYRK1ACDC7PLK4CHEK1
SCHEMBL1126627 0.75 HTT (0.45) HTTKDM4ECDK1MAPK1GSK3A
SCHEMBL1127274 0.74 HTT (0.44) HTTKDM4EDYRK1ACDC7PLK4
SCHEMBL1126791 0.74 HTT (0.44) HTTADRB2DYRK1ACDC7PLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2283006-A1 PYRROLE ANTIFUNGAL AGENTS F2G Limited (GB) 2011-02-16 EP disclosed
WO-2009130481-A1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2009-10-29 WO disclosed