SCHEMBL1127180

SCHEMBL1127180

COCCc1c(-c2ccccc2)c[nH]c1C=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 3/20 0.40
KDM4E B2RXH2 4/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
HTT P42858 1/20 0.38
ALDH1A1 P00352 2/20 0.35
RAB9A P51151 1/20 0.35
PARP1 P09874 1/20 0.35
GAA P10253 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CDC7 O00311 1/20 0.33
PLK4 O00444 1/20 0.33
CHEK1 O14757 1/20 0.33
CHUK O15111 1/20 0.33
PDPK1 O15530 1/20 0.33
DYRK3 O43781 1/20 0.33
ROCK2 O75116 1/20 0.33
PRKD3 O94806 1/20 0.33
MAP4K4 O95819 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1127247 0.79 HTT (0.48) ADRB2KDM4EL3MBTL1HTTALDH1A1
SCHEMBL1127088 0.72 HTT (0.47) ADRB2KDM4EL3MBTL1HTTALDH1A1
SCHEMBL1127206 0.71 HTT (0.46) ADRB2KDM4EL3MBTL1HTTALDH1A1
SCHEMBL5534778 0.70 ALDH1A1 (0.47) HTTALDH1A1RAB9APARP1SMN1; SMN2
SCHEMBL17800969 0.66 CD274 (0.43) ADRB2KDM4EL3MBTL1ALDH1A1RAB9A
SCHEMBL1126705 0.66 HTT (0.50) ADRB2KDM4EHTTALDH1A1RAB9A
SCHEMBL1127151 0.66 HTT (0.43) HTTALDH1A1PARP1CDC7PLK4
SCHEMBL28025320 0.65 ADRB2 (0.39) ADRB2KDM4EL3MBTL1HTTALDH1A1
SCHEMBL28451431 0.65 HTT (0.45) KDM4EHTTALDH1A1RAB9APARP1
SCHEMBL1126842 0.65 HTT (0.42) KDM4EHTTALDH1A1RAB9APARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2283006-A1 PYRROLE ANTIFUNGAL AGENTS F2G Limited (GB) 2011-02-16 EP disclosed
WO-2009130481-A1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2009-10-29 WO disclosed