SCHEMBL11273634

SCHEMBL11273634

COc1ccc2ccc(CC#N)cc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.50
CYP2A6 P11509 1/20 0.50
PTGS1 P23219 1/20 0.50
AKR1C3 P42330 1/20 0.50
AKR1C2 P52895 1/20 0.50
RAB9A P51151 2/20 0.47
KDM4E B2RXH2 2/20 0.47
NPC1 O15118 1/20 0.47
LMNA P02545 1/20 0.47
TP53 P04637 1/20 0.47
CYP3A4 P08684 1/20 0.47
MAPT P10636 1/20 0.47
MAOA P21397 1/20 0.47
SLC6A2 P23975 1/20 0.47
SLC6A3 Q01959 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
PTGS2 P35354 1/20 0.47
NQO1 P15559 1/20 0.46
PKM P14618 1/20 0.44
RAD52 P43351 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1448749 0.96 PTGS1 (0.53) CYP1A2CYP2A6PTGS1AKR1C3AKR1C2
SCHEMBL11272789 0.84 CYP1A2 (0.51) CYP1A2RAB9AKDM4ENPC1PKM
SCHEMBL6561661 0.81 KDM4E (0.59) CYP1A2CYP2A6KDM4ENPC1LMNA
SCHEMBL13970023 0.80 PTGS1 (0.47) CYP1A2CYP2A6PTGS1AKR1C3AKR1C2
SCHEMBL8538723 0.79 GLA (0.44) CYP1A2AKR1C3AKR1C2RAB9AKDM4E
SCHEMBL9428551 0.79 CYP1A2 (0.55) CYP1A2CYP2A6PTGS1AKR1C3AKR1C2
3-Methoxyphenylacetonitrile SCHEMBL103029 0.79 PKM (0.61) RAB9ANPC1LMNATP53CYP3A4
SCHEMBL11266053 0.79 PIK3CD (0.40) CYP1A2PTGS1AKR1C3AKR1C2RAB9A
SCHEMBL10424390 0.79 PTGS1 (0.57) CYP1A2CYP2A6PTGS1AKR1C3AKR1C2
SCHEMBL2222717 0.78 CYP1A2 (0.61) CYP1A2CYP2A6PTGS1AKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4327022-A Heterocyclic alkyl naphthols STERLING DRUG INC. (US) 1982-04-27 US disclosed
US-4169108-A 5(OR 6)-[(Substituted-amino)alkyl]-2,3-naphthalenediols STERLING DRUG INC. (US) 1979-09-25 US disclosed