SCHEMBL11266053

SCHEMBL11266053

COc1cc(OC)c2cc(CC#N)ccc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.40
PIK3CA P42336 1/20 0.40
PIK3CB P42338 1/20 0.40
PIK3CG P48736 1/20 0.40
PKM P14618 1/20 0.39
CYP1A2 P05177 2/20 0.38
PDE10A Q9Y233 2/20 0.37
TUBB4A P04350 1/20 0.37
TUBB P07437 1/20 0.37
TUBA3C P0DPH7 1/20 0.37
TUBA1B P68363 1/20 0.37
TUBA4A P68366 1/20 0.37
TUBB4B P68371 1/20 0.37
TUBB3 Q13509 1/20 0.37
TUBB2A Q13885 1/20 0.37
TUBB8 Q3ZCM7 1/20 0.37
TUBA3E Q6PEY2 1/20 0.37
TUBA1A Q71U36 1/20 0.37
TUBA1C Q9BQE3 1/20 0.37
TUBB6 Q9BUF5 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1448749 0.82 PTGS1 (0.53) PKMCYP1A2PDE10APTGDRKDM4E
SCHEMBL6944394 0.81 KDM4E (0.47) PIK3CDPIK3CAPIK3CBPIK3CGCYP1A2
SCHEMBL11276685 0.81 TTR (0.46) CYP1A2PDE10ATUBB4ATUBBTUBA3C
SCHEMBL11271678 0.81 CYP11B1 (0.42) CYP1A2PDE10ATUBB4ATUBBTUBA3C
SCHEMBL11272789 0.80 CYP1A2 (0.51) PIK3CDPIK3CAPIK3CBPIK3CGPKM
SCHEMBL11273634 0.79 CYP1A2 (0.50) PKMCYP1A2PDE10APTGDRKDM4E
SCHEMBL11471488 0.76 PTGS1 (0.68) KDM4ETDP1ALDH1A1HSD17B10NPC1
SCHEMBL77974 0.74 CA2 (0.61) PIK3CDPIK3CAPIK3CBPIK3CGCYP1A2
SCHEMBL6561661 0.73 KDM4E (0.59) CYP1A2KDM4ETDP1NPC1L3MBTL1
SCHEMBL12900679 0.72 ALDH1A1 (0.40) CYP1A2KDM4EALDH1A1CYP3A4HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4327022-A Heterocyclic alkyl naphthols STERLING DRUG INC. (US) 1982-04-27 US disclosed
US-4169108-A 5(OR 6)-[(Substituted-amino)alkyl]-2,3-naphthalenediols STERLING DRUG INC. (US) 1979-09-25 US disclosed