SCHEMBL11273639

SCHEMBL11273639

CCOc1nnc(-c2ccccc2)c(-c2ccccc2)n1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 1/20 0.49
NPSR1 Q6W5P4 1/20 0.47
ADORA2A P29274 4/20 0.47
ADORA1 P30542 4/20 0.47
LMNA P02545 2/20 0.46
TSHR P16473 1/20 0.46
ALDH1A1 P00352 4/20 0.45
SCN9A Q15858 1/20 0.45
HPGD P15428 2/20 0.44
RECQL P46063 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.43
KDM4E B2RXH2 2/20 0.43
GAA P10253 2/20 0.43
SQOR Q9Y6N5 1/20 0.43
CACNA2D1 P54289 1/20 0.43
NPC1 O15118 1/20 0.42
TP53 P04637 1/20 0.42
RAB9A P51151 1/20 0.42
ADORA2B P29275 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11483014 0.84 NQO1 (0.48) NPSR1LMNAALDH1A1SCN9AHPGD
SCHEMBL11239685 0.81 PTGES (0.50) GPR84NPSR1LMNAALDH1A1SCN9A
SCHEMBL11468702 0.81 TP53 (0.49) NPSR1LMNAALDH1A1SCN9AHPGD
SCHEMBL11244627 0.80 ADK (0.38) NPSR1TSHRALDH1A1SCN9AHPGD
SCHEMBL28303870 0.79 ADORA2A (0.52) GPR84NPSR1ADORA2AADORA1LMNA
SCHEMBL11268851 0.79 SMN1; SMN2 (0.53) GPR84NPSR1ADORA2AADORA1LMNA
SCHEMBL31582507 0.79 HTR7 (0.49) NPSR1ADORA2AADORA1LMNATSHR
SCHEMBL11469963 0.79 GAA (0.48) TSHRALDH1A1SCN9AHPGDSMN1; SMN2
SCHEMBL11471319 0.79 MAPT (0.37) NPSR1LMNATSHRALDH1A1SCN9A
SCHEMBL11467215 0.78 SCN9A (0.40) NPSR1ADORA2AADORA1LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4310551-A Pharmacologically active substituted 1,2,4-triazines DIAMOND SHAMROCK CORPORATION (US) 1982-01-12 US disclosed
US-4251527-A ANTIINFLAMMATORY AGENTS DIAMOND SHAMROCK CORPORATION (US) 1981-02-17 US disclosed
US-4157392-A HYPOTENSIVE AGENTS, ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIPYRETICS AND NERVOUS SYSTEM EFFECTS DIAMOND SHAMROCK CORPORATION (US) 1979-06-05 US disclosed