SCHEMBL11274121

SCHEMBL11274121

O=C(CBr)Nc1ccc(C2CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 2/20 0.53
HDAC11 Q96DB2 2/20 0.53
HDAC8 Q9BY41 2/20 0.53
HDAC6 Q9UBN7 2/20 0.53
MITF O75030 1/20 0.52
KLF5 Q13887 1/20 0.52
ALDH1A1 P00352 5/20 0.51
HPGD P15428 2/20 0.51
IDO1 P14902 1/20 0.51
NPC1 O15118 3/20 0.49
USP2 O75604 1/20 0.49
KMT2A Q03164 2/20 0.46
RAB9A P51151 2/20 0.46
RORC P51449 1/20 0.46
DEGS1 O15121 1/20 0.45
MEN1 O00255 1/20 0.44
TP53 P04637 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
SLC18A3 Q16572 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7735911 0.92 MITF (0.63) HDAC3HDAC11HDAC8HDAC6MITF
SCHEMBL15267699 0.82 KMT2A (0.60) HDAC3HDAC11HDAC8HDAC6MITF
SCHEMBL11272129 0.78 CA12 (0.56) HDAC3HDAC11HDAC8HDAC6MITF
SCHEMBL17361644 0.78 HPGD (0.61) HDAC3HDAC11HDAC8HDAC6MITF
SCHEMBL13242331 0.76 DGAT1 (0.51) IDO1NPC1RAB9ATP53SMN1; SMN2
SCHEMBL5868999 0.76 SLC18A3 (0.63) HDAC3HDAC11HDAC8HDAC6ALDH1A1
SCHEMBL12810977 0.76 HDAC3 (0.57) HDAC3HDAC11HDAC8HDAC6MITF
SCHEMBL1039601 0.75 KMT2A (0.76) ALDH1A1HPGDNPC1KMT2ARAB9A
SCHEMBL7888049 0.75 CYP1A1 (0.60) ALDH1A1HPGDNPC1KMT2ARAB9A
SCHEMBL517540 0.75 MITF (0.63) HDAC3HDAC11HDAC8HDAC6MITF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4348396-A Substituted 11-oxo-11H-pyrido[2,1-b]quinazolines and method of inhibiting allergic reactions with them HOFFMANN-LA ROCHE INC. (US) 1982-09-07 US disclosed