SCHEMBL11275455

SCHEMBL11275455

C=CCN(CCC)C1CCc2c[nH]cc2C1

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 1/20 0.61
HTR1B P28222 1/20 0.56
HTR1A P08908 2/20 0.51
DRD2 P14416 8/20 0.49
DRD3 P35462 7/20 0.49
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
CYP2D6 P10635 2/20 0.49
CYP1A2 P05177 2/20 0.49
TSHR P16473 2/20 0.49
ALDH1A1 P00352 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
FYN P06241 1/20 0.49
DRD4 P21917 2/20 0.46
ADRB2 P07550 1/20 0.46
CASP1 P29466 1/20 0.46
KDM4E B2RXH2 1/20 0.46
CYP3A4 P08684 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11267287 0.88 HTR1A (0.64) HTR1DHTR1BHTR1ADRD2DRD3
SCHEMBL11500383 0.86 HTR1D (0.47) HTR1DHTR1BHTR1ADRD2DRD3
Maleic Acid SCHEMBL11280479 0.84 ALDH1A1 (0.56) HTR1DHTR1BHTR1ADRD2DRD3
SCHEMBL2599107 0.83 HTR1A (0.76) HTR1DHTR1BHTR1ADRD2DRD3
SCHEMBL2599112 0.83 HTR1A (0.76) HTR1DHTR1BHTR1ADRD2DRD3
Sulfuric Acid SCHEMBL11263748 0.81 HTR1D (0.41) HTR1DHTR1BHTR1ADRD2DRD3
SCHEMBL11269661 0.80 SIGMAR1 (0.42) HTR1DHTR1BDRD2DRD3DRD4
SCHEMBL11268179 0.79 DRD2 (0.50) HTR1ADRD2DRD3MEN1KMT2A
SCHEMBL8315256 0.76 HTR1D (1.00) HTR1DHTR1B
Hydrochloric Acid SCHEMBL9752128 0.75 DRD3 (0.59) HTR1DHTR1BHTR1ADRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0014792-B1 TETRAHYDRO-2H-BENZO(C)PYRROLES, THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THE COMPOUNDS FOR USE AS THERAPEUTICALS ELI LILLY AND COMPANY (US) 1982-12-01 EP disclosed
US-4264622-A TREATMENT OF PARKINSON*S DISEASE ELI LILLY AND COMPANY (US) 1981-04-28 US disclosed
US-4235776-A USED FOR TREATMENT OF PARKINSON'S DISEASE, PROLACTIN INHIBITORS, AND DOPAMINE AGONISTS ELI LILLY AND COMPANY (US) 1980-11-25 US disclosed