SCHEMBL11277959

SCHEMBL11277959

O=C(O)CN(Cc1ccccc1)C(=O)CCS

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.46
RAB9A P51151 2/20 0.46
ALOX5 P09917 2/20 0.45
LMNA P02545 2/20 0.45
TSHR P16473 2/20 0.44
ESR1 P03372 1/20 0.44
POLB P06746 1/20 0.44
NR4A1 P22736 1/20 0.44
ALOX15 P16050 1/20 0.44
MAPK1 P28482 1/20 0.44
HSD17B10 Q99714 1/20 0.44
ALDH1A1 P00352 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
REN P00797 1/20 0.43
KMT2A Q03164 1/20 0.42
AGTR1 P30556 1/20 0.42
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC10 Q969S8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3125812 0.90 NPC1 (0.52) NPC1RAB9AALOX5LMNATSHR
SCHEMBL6314236 0.84 LMNA (0.49) NPC1RAB9AALOX5LMNATSHR
SCHEMBL6314244 0.81 LMNA (0.49) NPC1RAB9AALOX5LMNATSHR
SCHEMBL19567152 0.80 CTSL (0.49) NPC1RAB9ALMNATSHRESR1
SCHEMBL7301929 0.80 LMNA (0.55) NPC1RAB9ALMNATSHRMAPK1
SCHEMBL18666669 0.78 ACE (0.42) LMNATSHRALOX15ACE
SCHEMBL3750325 0.77 POLB (0.59) NPC1RAB9AALOX5LMNATSHR
SCHEMBL3130089 0.77 NPC1 (0.53) NPC1RAB9AALOX5LMNATSHR
SCHEMBL11271784 0.76 HDAC1 (0.43) NPC1RAB9AALOX5LMNATSHR
SCHEMBL8465299 0.76 MAPK1 (0.54) NPC1ALOX5LMNATSHRALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4339600-A ENZYME INHIBITORS E. R. SQUIBB & SONS, INC. (US) 1982-07-13 US disclosed
US-4199512-A Compounds for alleviating hypertension E. R. SQUIBB & SONS, INC. (US) 1980-04-22 US disclosed
US-4173704-A HYPOTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1979-11-06 US disclosed
US-4140786-A ENZYME INHIBITORS E. R. SQUIBB & SONS, INC. (US) 1979-02-20 US disclosed
US-4140797-A MERCAPTOACYL AMINO ACIDS, ENZYME INHIBITORS E. R. SQUIBB & SONS, INC. (US) 1979-02-20 US disclosed
US-4112119-A MERCAPTOACYL AMINOACIDS E. R. SQUIBB & SONS, INC. (US) 1978-09-05 US disclosed
US-4053651-A MERCAPTOACYL AMINO ACIDS, ENZYME INHIBITORS E. R. SQUIBB & SONS, INC. (US) 1977-10-11 US disclosed