SCHEMBL11277987

SCHEMBL11277987

Cc1cc(Cl)cc(Cl)c1N(C)C(=O)NC(=N)N

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.34
FSCN1 Q16658 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
HTR3E A5X5Y0 1/20 0.33
HTR3B O95264 1/20 0.33
HTR3A P46098 1/20 0.33
HTR3D Q70Z44 1/20 0.33
HTR3C Q8WXA8 1/20 0.33
APEX1 P27695 1/20 0.33
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
RAPGEF4 Q8WZA2 1/20 0.32
ABCB1 P08183 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
F2 P00734 1/20 0.30
ALDH1A1 P00352 2/20 0.30
MAPT P10636 2/20 0.30
GAA P10253 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11269830 0.99 KDM4E (0.33) KDM4EFSCN1TDP1HTR3EHTR3B
SCHEMBL11414012 0.92 HTR3E (0.35) KDM4EHTR3EHTR3BHTR3AHTR3D
SCHEMBL11320156 0.92 FSCN1 (0.36) KDM4EFSCN1HTR3EHTR3BHTR3A
SCHEMBL11404870 0.88 HTT (0.37) KDM4ERAB9AL3MBTL1CA1CA2
SCHEMBL11422730 0.86 FSCN1 (0.32) KDM4EFSCN1HTR3EHTR3BHTR3A
SCHEMBL11405232 0.86 BDKRB1 (0.31) KDM4EHTR3EHTR3BHTR3AHTR3D
SCHEMBL11430940 0.86 CA1 (0.32) FSCN1HTR3EHTR3BHTR3AHTR3D
SCHEMBL11419163 0.86 CA1 (0.32) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL11277637 0.86 ALDH1A1 (0.32) KDM4ECA1CA2ALDH1A1MAPK1
SCHEMBL11406819 0.85 HTR3E (0.34) KDM4EHTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4150154-A GASTROINTESTINAL ANTISPASMODICS WILLIAM H. RORER, INC. (US) 1979-04-17 US claimed
US-4326075-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4283555-A Amidinoureas WILLIAM H. RORER, INC. (US) 1981-08-11 US disclosed
US-4219567-A ANTIULCER AGENTS WILLIAM H. RORER, INC. (US) 1980-08-26 US disclosed
US-4216229-A 1-AMIDINO-3-PHENYLUREAS WILLIAM H. RORER, INC. (US) 1980-08-05 US disclosed
US-4216230-A Method for alleviating hypertension with amidinoureas WILLIAM H. RORER, INC. (US) 1980-08-05 US disclosed
US-4203920-A ANTIDIARRHEAL WILLIAM H. RORER, INC. (US) 1980-05-20 US disclosed
US-4183956-A Method for treating gastrointestinal spasms, gastrointestinal hyperacidity and hypertensive disorders with amidinoureas WILLIAM H. RORER, INC. (US) 1980-01-15 US disclosed
US-4150154-A GASTROINTESTINAL ANTISPASMODICS WILLIAM H. RORER, INC. (US) 1979-04-17 US disclosed
US-4060635-A Amidinoureas for treating diarrhea WILLIAM H. RORER, INC. (US) 1977-11-29 US disclosed