SCHEMBL11052411

SCHEMBL11052411

CNC(=N)NC(=O)Nc1c(C)cc(Br)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.41
TSHR P16473 1/20 0.41
ALDH1A1 P00352 7/20 0.40
MAPT P10636 2/20 0.40
KMT2A Q03164 2/20 0.40
LMNA P02545 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
HPGD P15428 2/20 0.38
POLB P06746 2/20 0.38
IDH1 O75874 1/20 0.38
MEN1 O00255 1/20 0.36
RAB9A P51151 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
TAS1R2 Q8TE23 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11134528 0.99 HTT (0.40) HTTTSHRALDH1A1MAPTKMT2A
SCHEMBL11285813 0.87 HTT (0.38) HTTTSHRALDH1A1MAPTKMT2A
SCHEMBL11279723 0.84 HTT (0.42) HTTTSHRALDH1A1MAPTKMT2A
Hydrochloric Acid SCHEMBL11080185 0.84 HTT (0.38) HTTTSHRALDH1A1MAPTKMT2A
SCHEMBL11054649 0.84 SCN5A (0.35) HTTTSHRALDH1A1MAPTKMT2A
SCHEMBL11810046 0.77 ALDH1A1 (0.31) ALDH1A1
SCHEMBL11051094 0.77 ALDH1A1 (0.58) ALDH1A1KMT2ALMNAHPGDPOLB
SCHEMBL10612997 0.77 PDK1 (0.48) POLBIDH1
SCHEMBL10907930 0.76 ALDH1A1 (0.43) ALDH1A1KMT2ALMNAPOLBMEN1
Hydrochloric Acid SCHEMBL11505921 0.76 PKM (0.48) POLBIDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4326075-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed
US-4203920-A ANTIDIARRHEAL WILLIAM H. RORER, INC. (US) 1980-05-20 US disclosed
US-4147804-A ANTIARRHYTHMIA AGENTS WILLIAM H. RORER, INC. (US) 1979-04-03 US disclosed
US-4060635-A Amidinoureas for treating diarrhea WILLIAM H. RORER, INC. (US) 1977-11-29 US disclosed