SCHEMBL11289808

SCHEMBL11289808

CC(=O)C1=CC2(CCCC2)c2ccccc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 6/20 0.37
AKR1C1 Q04828 1/20 0.37
NOTUM Q6P988 2/20 0.36
THRB P10828 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
PDK2 Q15119 2/20 0.34
GAA P10253 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
KMT2A Q03164 2/20 0.33
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 2/20 0.33
MAPT P10636 2/20 0.33
HTT P42858 1/20 0.33
APAF1 O14727 1/20 0.33
TDP2 O95551 1/20 0.33
NSD2 O96028 1/20 0.33
RECQL P46063 1/20 0.33
SAE1 Q9UBE0 1/20 0.33
UBA2 Q9UBT2 1/20 0.33
NPC1 O15118 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11292902 0.80 HDAC4 (0.33) HDAC4AKR1C1THRBTDP1PDK2
SCHEMBL11287867 0.80 PTPN1 (0.37) HDAC4AKR1C1THRBTDP1PDK2
SCHEMBL11290184 0.79 KDM4E (0.38) HDAC4AKR1C1PDK2SMN1; SMN2KMT2A
SCHEMBL11544999 0.72 AKR1C1 (0.37) HDAC4AKR1C1THRBTDP1PDK2
SCHEMBL3539163 0.71 OPRD1 (0.40) THRBTDP1SMN1; SMN2ALDH1A1HPGD
SCHEMBL4006116 0.71 SCN1A (0.39) NOTUMPDK2KMT2AKDM4EGLA
SCHEMBL11295881 0.71 PGR (0.33) HDAC4AKR1C1ALDH1A1KDM4E
SCHEMBL3538240 0.70 OPRD1 (0.45) PDK2GAASMN1; SMN2ALDH1A1KDM4E
SCHEMBL11290237 0.69 PGR (0.35) HDAC4ALDH1A1KDM4E
SCHEMBL11294472 0.69 HDAC4 (0.35) HDAC4PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0000825-B1 GEMINALLY DISUBSTITUTED INDENE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Kabi AB (SE) 1982-04-14 EP disclosed
US-4218472-A USED AS DECONGESANT, HYPOTENSIVE AGENT, VASOCONSTRICTOR, ANTI-RESERPINE AGENT, TREATING INCONTINENCE AB KABI (SE) 1980-08-19 US disclosed
EP-0000825-A1 Geminally disubstituted indene derivatives, processes for their preparation and pharmaceutical compositions containing them Kabi AB (SE) 1979-02-21 EP disclosed