SCHEMBL11290237

SCHEMBL11290237

BrC1=CC2(CCCCC2)c2ccccc21

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PGR P06401 3/20 0.35
HDAC4 P56524 1/20 0.33
PDE7A Q13946 3/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11295881 0.98 PGR (0.33) PGRHDAC4KDM4EALDH1A1
SCHEMBL11289903 0.90 S100A4 (0.33) ALDH1A1
SCHEMBL11354579 0.74 PGR (0.35) PGRHDAC4PDE7AALDH1A1
SCHEMBL11544758 0.73 SLC6A3 (0.42)
SCHEMBL9441510 0.72 PDK2 (0.37) PGR
SCHEMBL11544153 0.72
SCHEMBL11292078 0.72 PGR (0.33) PGRPDE7A
SCHEMBL11287867 0.70 PTPN1 (0.37) HDAC4
SCHEMBL11289410 0.70
SCHEMBL30913188 0.69 MEN1 (0.38) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0000825-B1 GEMINALLY DISUBSTITUTED INDENE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Kabi AB (SE) 1982-04-14 EP disclosed
US-4218472-A USED AS DECONGESANT, HYPOTENSIVE AGENT, VASOCONSTRICTOR, ANTI-RESERPINE AGENT, TREATING INCONTINENCE AB KABI (SE) 1980-08-19 US disclosed
EP-0000825-A1 Geminally disubstituted indene derivatives, processes for their preparation and pharmaceutical compositions containing them Kabi AB (SE) 1979-02-21 EP disclosed