SCHEMBL11295489

SCHEMBL11295489

Nc1cc(F)c(N2CCNCC2)cc1F

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
MAPT P10636 3/20 0.48
LMNA P02545 2/20 0.48
GAA P10253 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.47
OPRL1 P41146 2/20 0.44
NCF1 P14598 1/20 0.40
HRH4 Q9H3N8 1/20 0.40
SMARCA2 P51531 1/20 0.39
SMARCA4 P51532 1/20 0.39
PBRM1 Q86U86 1/20 0.39
HTR7 P34969 2/20 0.39
ADRB1 P08588 2/20 0.39
KDR P35968 1/20 0.38
HTR1A P08908 1/20 0.38
HTR2B P41595 1/20 0.38
HTR3A P46098 1/20 0.38
HTR6 P50406 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8070794 0.91 ALDH1A1 (0.51) ALDH1A1MAPTLMNAGAASMN1; SMN2
SCHEMBL7544806 0.84 ALDH1A1 (0.61) ALDH1A1MAPTLMNAGAASMN1; SMN2
SCHEMBL11296687 0.84 HTR3A (0.46) ALDH1A1MAPTLMNAGAAOPRL1
SCHEMBL6582872 0.84 ALDH1A1 (0.56) ALDH1A1MAPTLMNAGAASMN1; SMN2
Tert-Butyl Formate SCHEMBL27944987 0.82 MAPT (0.39) ALDH1A1MAPTLMNAGAASMN1; SMN2
SCHEMBL27046957 0.82 HTR3E (0.51) ALDH1A1MAPTLMNAGAAOPRL1
SCHEMBL29728648 0.81 ALDH1A1 (0.53) ALDH1A1MAPTLMNAGAASMN1; SMN2
SCHEMBL238269 0.81 ALDH1A1 (0.53) ALDH1A1MAPTLMNAGAASMN1; SMN2
SCHEMBL24632626 0.78 ADRB1 (0.50) ALDH1A1MAPTLMNAGAASMN1; SMN2
SCHEMBL16514396 0.78 ALDH1A1 (0.57) ALDH1A1MAPTLMNAGAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2665727-A1 BICYCLIC CARBOXAMIDE INHIBITORS OF KINASES Abbvie Inc. (US) 2013-11-27 EP disclosed
EP-2665724-A1 BICYCLIC INHIBITORS OF ALK AbbVie Inc. (US) 2013-11-27 EP disclosed
WO-2012097684-A1 BICYCLIC CARBOXAMIDE INHIBITORS OF KINASES ABBOTT LABORATORIES (US) 2012-07-26 WO disclosed
WO-2012097682-A1 BICYCLIC INHIBITORS OF ALK ABBOTT LABORATORIES (US) 2012-07-26 WO disclosed