SCHEMBL11298161

SCHEMBL11298161

CCCC(C)C(=O)NC1CCc2cccc(N)c2C1

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 11/20 0.54
MTNR1B P49286 11/20 0.54
CYP1A2 P05177 1/20 0.48
MAPT P10636 1/20 0.48
CYP2C9 P11712 1/20 0.48
ALOX15 P16050 1/20 0.48
TAOK1 Q7L7X3 3/20 0.42
TAOK3 Q9H2K8 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11294282 0.83 MTNR1A (0.64) MTNR1AMTNR1BTAOK1TAOK3
SCHEMBL8885912 0.76 CA1 (0.40) MTNR1AMTNR1BTAOK1TAOK3
SCHEMBL6561215 0.76 GRM7 (0.60) MTNR1AMTNR1BMAPTTAOK1TAOK3
SCHEMBL9759525 0.74 DRD2 (0.43) MTNR1AMTNR1BCYP1A2MAPTCYP2C9
SCHEMBL1965788 0.74 MTNR1A (0.52) MTNR1AMTNR1BCYP1A2MAPTCYP2C9
SCHEMBL8887633 0.74 HTR1D (0.57) MTNR1AMTNR1BTAOK1TAOK3
SCHEMBL9758631 0.73 MTNR1A (0.41) MTNR1AMTNR1BCYP1A2MAPTCYP2C9
SCHEMBL9241335 0.72 MTNR1A (0.68) MTNR1AMTNR1BCYP1A2MAPTCYP2C9
Hydrochloric Acid SCHEMBL9242722 0.72 MTNR1A (0.67) MTNR1AMTNR1BCYP1A2MAPTCYP2C9
Hydrochloric Acid SCHEMBL9243601 0.72 MTNR1A (0.67) MTNR1AMTNR1BCYP1A2MAPTCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1981003491-A1 THERAPEUTICALLY USEFUL TETRALIN DERIVATIVES ASTRA LAEKEMEDEL AB (SE) 1981-12-10 WO disclosed
EP-0041488-A1 Therapeutically useful tetralin derivatives Arvidsson, Folke Lars-Erik (SE) 1981-12-09 EP disclosed