SCHEMBL8887633

SCHEMBL8887633

CCCC(C)C(=O)NC1CCc2cc(F)ccc2C1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 1/20 0.57
HTR1B P28222 1/20 0.57
PSEN1 P49768 1/20 0.47
PSEN2 P49810 1/20 0.47
APH1B Q8WW43 1/20 0.47
NCSTN Q92542 1/20 0.47
APH1A Q96BI3 1/20 0.47
PSENEN Q9NZ42 1/20 0.47
MTNR1A P48039 5/20 0.45
MTNR1B P49286 5/20 0.45
PRMT5 O14744 2/20 0.45
GRM7 Q14831 1/20 0.44
CA1 P00915 4/20 0.44
CA2 P00918 4/20 0.44
CA12 O43570 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
ACHE P22303 2/20 0.44
TAOK1 Q7L7X3 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11294282 0.84 MTNR1A (0.64) MTNR1AMTNR1BGRM7TAOK1TAOK3
SCHEMBL8885912 0.82 CA1 (0.40) HTR1DHTR1BMTNR1AMTNR1BCA1
SCHEMBL5121715 0.79 HTR1D (0.60) HTR1DHTR1BPSEN1PSEN2APH1B
SCHEMBL5121719 0.79 HTR1D (0.60) HTR1DHTR1BPSEN1PSEN2APH1B
SCHEMBL2819567 0.79 HTR1D (0.60) HTR1DHTR1BPSEN1PSEN2APH1B
SCHEMBL8884861 0.78 GAA (0.43) HTR1DHTR1BMTNR1AMTNR1BCA1
SCHEMBL6561215 0.77 GRM7 (0.60) MTNR1AMTNR1BGRM7CA1CA2
SCHEMBL6932016 0.76 MTNR1A (0.38) MTNR1AMTNR1BCA1CA2CA12
SCHEMBL6561214 0.76 CA1 (0.56) GRM7CA1CA2CA12CA7
SCHEMBL11298161 0.74 MTNR1A (0.54) MTNR1AMTNR1BTAOK1TAOK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5650427-A ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1997-07-22 US disclosed
US-5461061-A Antidepressants WIKSTROM HAKAN V (NL) 1995-10-24 US disclosed
US-5288748-A Antidepressants THE UPJOHN COMPANY (US) 1994-02-22 US disclosed
EP-0510068-A1 NEW CENTRALLY ACTING 6,7,8,9-TETRAHYDRO-3H-BENZ(e)INDOLE HETEROCYCLICS PHARMACIA & UPJOHN COMPANY (US) 1992-10-28 EP disclosed
WO-1991011435-A2 NEW CENTRALLY ACTING 6,7,8,9-TETRAHYDRO-3H-BENZ(e)INDOLE HETEROCYCLICS THE UPJOHN COMPANY (US) 1991-08-08 WO disclosed