SCHEMBL11299758

SCHEMBL11299758

CCc1nc2sc(C)c(C)c2c(=O)n1OC(=O)NC

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAK O14976 1/20 0.56
MAPK1 P28482 2/20 0.45
ALDH1A1 P00352 4/20 0.44
GAA P10253 3/20 0.44
HPGD P15428 2/20 0.44
KDM4E B2RXH2 2/20 0.44
CYP1A2 P05177 1/20 0.44
POLB P06746 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
TSHR P16473 3/20 0.44
LMNA P02545 1/20 0.41
PKM P14618 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
USP2 O75604 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11301157 0.69 ALDH1A1 (0.47) GAKMAPK1ALDH1A1GAAHPGD
SCHEMBL11299230 0.68 GAK (0.57) GAKMAPK1ALDH1A1GAAHPGD
SCHEMBL11518343 0.61 KDM4E (0.71) MAPK1ALDH1A1GAAHPGDKDM4E
SCHEMBL12310881 0.59 ALDH1A1 (0.46) ALDH1A1GAAHPGDKDM4ECYP1A2
SCHEMBL7017261 0.59 MAPK1 (0.49) GAKMAPK1ALDH1A1GAAPOLB
SCHEMBL11485343 0.58 ELANE (0.60) ALDH1A1GAAHPGDKDM4ECYP1A2
SCHEMBL12892166 0.57 HTT (0.68) MAPK1ALDH1A1GAAPOLBLMNA
SCHEMBL5265815 0.57 ALDH1A1 (0.69) MAPK1ALDH1A1GAAHPGDKDM4E
SCHEMBL12877215 0.57 LMNA (0.79) MAPK1ALDH1A1HPGDKDM4EPOLB
SCHEMBL12261730 0.57 GAK (0.43) GAKMAPK1ALDH1A1GAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-56059778-A None JP disclosed
JP-S5659778-A DIMETHYLTHIENOPYRIMIDIONE DERIVATIVE SHOWA DENKO KK 1981-05-23 JP disclosed