SCHEMBL7017261

SCHEMBL7017261

Cc1sc2nc(S)n(C)c(=O)c2c1C

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.49
GAK O14976 1/20 0.49
TSHR P16473 2/20 0.48
ALDH1A1 P00352 4/20 0.47
USP2 O75604 2/20 0.47
LMNA P02545 2/20 0.47
HTT P42858 1/20 0.47
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.44
ATM Q13315 1/20 0.44
MEN1 O00255 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14360622 0.82 MAPT (0.54) MAPK1GAKTSHRALDH1A1USP2
SCHEMBL1101894 0.77 MAPK1 (0.60) MAPK1GAKTSHRALDH1A1USP2
SCHEMBL7018716 0.71 ERCC5 (0.41) MAPK1TSHRALDH1A1HTTGAA
SCHEMBL3754226 0.70 GAK (0.67) MAPK1GAKALDH1A1USP2LMNA
Potassium Ion SCHEMBL3689408 0.68 GAK (0.63) MAPK1GAKTSHRALDH1A1USP2
SCHEMBL7018863 0.67 KDM4E (0.33) ALDH1A1LMNAHTTNPC1RAB9A
SCHEMBL14478932 0.67 ALDH1A1 (0.63) MAPK1TSHRALDH1A1USP2LMNA
SCHEMBL12718463 0.64 MAPK1 (0.43) MAPK1GAKTSHRGAAMAPT
SCHEMBL11299230 0.64 GAK (0.57) MAPK1GAKTSHRALDH1A1USP2
SCHEMBL799433 0.63 ADORA2B (0.45) MAPK1TSHRALDH1A1USP2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836602-B1 FUNGICIDAL PYRIMIDINONES DU PONT (US) 2002-01-30 EP claimed
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-6348504-B1 COMPOUNDS WITH AMIDINE OR GUANIDINE GROUPS AND CARBOXY OR ESTER GROUPS THROMBOLYTICS AND/OR FOR THE TREATMENT OF THROMBOEMBOLIC DISORDERS. DUPONT PHARMACEUTICALS COMPANY 2002-02-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed