SCHEMBL11301435

SCHEMBL11301435

COc1cc(SC)ccc1-c1nc2ccc(C3(C)C=NNC(=O)C3)cc2[nH]1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 13/20 0.38
PDE5A O76074 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
CHEK2 O96017 1/20 0.35
NPC1 O15118 1/20 0.34
HSP90AA1 P07900 1/20 0.34
PKM P14618 1/20 0.34
RAB9A P51151 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
TP53 P04637 1/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11306274 0.88 AMY1A (0.43) AMY1APDE3BPDE3ANPC1PKM
Hydrochloric Acid SCHEMBL11307551 0.87 AMY1A (0.42) AMY1APDE3BPDE3ANPC1PKM
SCHEMBL7357180 0.85 AMY1A (0.37) AMY1APDE5APDE3BPDE3AHDAC6
SCHEMBL7356104 0.81 KDM4E (0.48) AMY1APDE3BPDE3ACHEK2MAPT
SCHEMBL7352154 0.80 ALDH1A1 (0.48) NPC1HSP90AA1RAB9AMAPT
SCHEMBL7348936 0.79 AURKA (0.42) AMY1APDE3BPDE3ACHEK2NPC1
SCHEMBL7357077 0.78 ABCB11 (0.52) PDE3BPDE3ACHEK2NPC1PKM
Hydrochloric Acid SCHEMBL11304721 0.78 ABCB11 (0.52) PDE3BPDE3ACHEK2NPC1PKM
SCHEMBL7347482 0.76 NPC1 (0.46) AMY1ANPC1PKMRAB9AHDAC6
SCHEMBL7350293 0.76 NPC1 (0.49) PDE3BPDE3ANPC1PKMRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4361563-A CARDIOTONIC, ANTITHROMBOTIC DR. KARL THOMAE GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1982-11-30 US disclosed