SCHEMBL11301733

SCHEMBL11301733

CCOc1cccc(C(=O)OC)c1O

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KLK1 P06870 1/20 0.53
KLK5 Q9Y337 1/20 0.53
HCRTR1 O43613 2/20 0.51
MAPT P10636 3/20 0.50
KCNK3 O14649 1/20 0.49
KCNK9 Q9NPC2 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
GAA P10253 1/20 0.49
MAPK1 P28482 1/20 0.49
LMNA P02545 2/20 0.49
TSHR P16473 1/20 0.49
L3MBTL1 Q9Y468 2/20 0.48
GRM5 P41594 1/20 0.48
HTT P42858 1/20 0.48
TAS1R3 Q7RTX0 1/20 0.48
TAS1R1 Q7RTX1 1/20 0.48
KMT2A Q03164 1/20 0.47
SLC6A3 Q01959 1/20 0.45
GLA P06280 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8108839 0.85 KLKB1 (0.49) KLK1KLK5LMNATSHRL3MBTL1
SCHEMBL30553984 0.84 HCRTR1 (0.65) HCRTR1MAPTKCNK3KCNK9TDP1
SCHEMBL1989129 0.84 HCRTR1 (0.65) HCRTR1MAPTKCNK3KCNK9TDP1
SCHEMBL21543727 0.83 HCRTR1 (0.51) HCRTR1MAPTKCNK3KCNK9TDP1
SCHEMBL9324858 0.83 LMNA (0.57) MAPTMAPK1LMNATSHRHTT
SCHEMBL8117696 0.83 KLK1 (0.56) KLK1KLK5HCRTR1MAPTKCNK3
SCHEMBL539003 0.83 KLK1 (0.52) KLK1KLK5HCRTR1MAPTGAA
Methyl 2-Hydroxy-3-Methoxybenzoate SCHEMBL1339162 0.82 TAS1R3 (0.56) KLK1KLK5MAPTGAAMAPK1
SCHEMBL24009066 0.82 ALDH1A1 (0.50) HCRTR1MAPTKCNK3KCNK9TDP1
SCHEMBL30288409 0.82 ALDH1A1 (0.50) HCRTR1MAPTKCNK3KCNK9TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0009780-B1 OCTAHYDRO-1H-BENZO(4,5)FURO(3,2-E)ISOQUINOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM E.I. DU PONT DE NEMOURS AND COMPANY (US) 1982-02-24 EP disclosed
US-4260761-A Intermediates for the preparation of octahydro-1H-benzo[4,5]furo[3,2,-e]-isoquinoline analgesic and narcotic antagonistic compounds E. I. DU PONT DE NEMOURS AND COMPANY (US) 1981-04-07 US disclosed
US-4243668-A Octahydro-1H-benzo[4,5]furo[3,2-e]-isoquinoline analgesic and narcotic antagonistic compounds E. I. DU PONT DE NEMOURS AND COMPANY (US) 1981-01-06 US disclosed
EP-0009780-A2 Octahydro-1H-benzo(4,5)furo(3,2-e)isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them E.I. DU PONT DE NEMOURS AND COMPANY (US) 1980-04-16 EP disclosed
US-4053415-A UNSATURATED POLYESTER ETHER HAVING A PHOTOCROSSLINKABLE MOIETY FUJI PHOTO FILM CO., LTD. (JA) 1977-10-11 US disclosed