SCHEMBL113065

SCHEMBL113065

COc1cc(OC)cc(C(C)COC(N)=O)c1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.44
TNF P01375 1/20 0.44
CYP1A2 P05177 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
CYP2D6 P10635 1/20 0.41
PKM P14618 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
KMT2A Q03164 2/20 0.40
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
MTNR1A P48039 3/20 0.36
MTNR1B P49286 3/20 0.36
ALOX5 P09917 1/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21465394 1.00 L3MBTL1 (0.44) L3MBTL1TNFCYP1A2SMN1; SMN2CYP2D6
SCHEMBL2452044 0.80 ABCB11 (0.61) L3MBTL1CYP1A2LMNAALOX5
SCHEMBL2452047 0.80 ABCB11 (0.61) L3MBTL1CYP1A2LMNAALOX5
SCHEMBL28958757 0.74 CYP1A2 (0.68) CYP1A2SMN1; SMN2CYP2D6PKMNPSR1
SCHEMBL4589554 0.74 CYP1A2 (0.68) CYP1A2SMN1; SMN2CYP2D6PKMNPSR1
SCHEMBL528282 0.74 KMT2A (0.43) L3MBTL1TNFCYP1A2KMT2AALDH1A1
SCHEMBL4590669 0.74 CYP1A2 (0.68) CYP1A2SMN1; SMN2CYP2D6PKMNPSR1
SCHEMBL5497954 0.72 ALDH1A1 (0.39) TNFKMT2AALDH1A1POLBMTNR1A
SCHEMBL5497959 0.72 ALDH1A1 (0.39) PKMKMT2AALDH1A1POLBMTNR1A
SCHEMBL14861206 0.72 L3MBTL1 (0.61) L3MBTL1CYP1A2SMN1; SMN2CYP2D6PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 426 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026107431-A1 STEREOSELECTIVE SYNTHESIS OF L,2-CIS-2-AMINOGLYCOSIDES BRANDEIS UNIVERSITY (US) 2026-05-21 WO disclosed
EP-4734976-A2 AGENTS FOR TREATING DISORDERS INVOLVING RYANODINE RECEPTORS RyCarma Therapeutics, Inc. (US) 2026-05-06 EP disclosed
WO-2026090589-A1 HETEROCYCLIC HBS1L DEGRADERS TANGO THERAPEUTICS, INC. (US) 2026-04-30 WO disclosed
EP-4688758-A1 VERDAZYL COMPOUNDS AS CONTRAST AGENTS FOR MAGNETIC RESONANCE IMAGING OF KIDNEYS Yellowbird Diagnostics Inc. (CA) 2026-02-11 EP disclosed
EP-4658280-A2 SIX MEMBERED RING CONTAINING OLIGOMERS Alnylam Pharmaceuticals, Inc. (US) 2025-12-10 EP disclosed
EP-4543990-A1 INDOCYANINE GREEN (ICG) MODIFICATION FOR TREATMENT OF LIVER CANCER The Children's Medical Center Corporation (US) 2025-04-30 EP disclosed
WO-2025006617-A2 AGENTS FOR TREATING DISORDERS INVOLVING RYANODINE RECEPTORS ARMGO PHARMA, INC. (US) 2025-01-02 WO disclosed
WO-2024220852-A2 TEAD CORE INHIBITORS FOR CANCER THERAPEUTICS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2024-10-24 WO disclosed
EP-4444274-A1 COMPOSITIONS COMPRISING MODIFIED PHOSPHOLIPIDS AND USES THEREOF The Children's Medical Center Corporation (US) 2024-10-16 EP disclosed
EP-4440560-A1 SMALL MOLECULE INHIBITORS OF REPEAT ASSOCIATED NON-AUG (RAN) TRANSLATION AND COMBINATION THERAPIES UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2024-10-09 EP disclosed
WO-2009020768-A1 TARGETING THE ONCOPROTEIN NUCLEOPHOSMIN PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2009-02-12 WO disclosed
WO-2009018088-A2 IMAGING OF ALPHA-SYNUCLEIN LINK MEDICINE CORPORATION (US) 2009-02-05 WO disclosed
WO-2008137692-A1 TREATMENT OF SYNUCLEINOPATHIES LINK MEDICINE CORPORATION (US) 2008-11-13 WO disclosed
WO-2008127361-A2 SYNTHESIS OF ENONE INTERMEDIATE PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2008-10-23 WO disclosed
WO-2008121767-A2 STITCHED POLYPEPTIDES PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2008-10-09 WO disclosed
WO-2008122038-A1 REGULATING AUTOPHAGY PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2008-10-09 WO disclosed
WO-2008119015-A2 SYNTHESIS OF THIOHYDANTOINS SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 2008-10-02 WO disclosed
WO-2008063300-A2 BORONIC ACIDS AND ESTERS AS INHIBITORS OF FATTY ACID AMIDE HYDROLASE INFINITY PHARMACEUTICALS, INC. (US) 2008-05-29 WO disclosed
EP-0970066-A1 AMINOEPOXIDES FROM AMINOALDEHYDES AND IN-SITU FORMED HALOMETHYL ORGANOMETALLIC REAGENT G.D. SEARLE & CO. (US) 2000-01-12 EP disclosed
WO-1998029401-A1 AMINOEPOXIDES FROM AMINOALDEHYDES AND IN-SITU FORMED HALOMETHYL ORGANOMETALLIC REAGENT G.D. SEARLE & CO. (US) 1998-07-09 WO disclosed