SCHEMBL11333344

SCHEMBL11333344

Cc1cc(OCC(O)CNC(C)C)c2[nH]c(=S)[nH]c2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.51
DRD3 P35462 2/20 0.51
ABCB11 O95342 1/20 0.51
ADRA2A P08913 1/20 0.51
PTGS1 P23219 1/20 0.51
SLC6A2 P23975 1/20 0.51
OPRM1 P35372 1/20 0.51
ADRB2 P07550 6/20 0.48
ADRB1 P08588 6/20 0.48
ADRB3 P13945 3/20 0.48
DNM1 Q05193 1/20 0.46
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 2/20 0.45
LMNA P02545 2/20 0.45
KDM4E B2RXH2 1/20 0.45
USP2 O75604 1/20 0.45
CYP2D6 P10635 1/20 0.45
THRB P10828 1/20 0.45
CYP2C9 P11712 1/20 0.45
TSHR P16473 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11184202 0.86 HTR1A (0.51) HTR1ADRD3ABCB11ADRA2APTGS1
SCHEMBL11352195 0.85 MAPT (0.52) ADRB2ADRB1ADRB3CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL11185783 0.85 ADRB2 (0.51) HTR1ADRD3ABCB11ADRA2APTGS1
Hydrochloric Acid SCHEMBL11377640 0.84 MAPT (0.54) ADRB2ADRB1ADRB3CYP1A2CYP3A4
SCHEMBL11468630 0.82 ADRB2 (0.63) HTR1ADRD3ABCB11ADRA2APTGS1
SCHEMBL11449996 0.75 ADRB2 (0.70) HTR1ADRD3ABCB11ADRA2APTGS1
SCHEMBL13495721 0.74 ADRB2 (0.76) HTR1ADRD3ABCB11ADRA2APTGS1
SCHEMBL11460105 0.73 ABCB11 (0.51) HTR1ADRD3ABCB11ADRA2APTGS1
SCHEMBL11861389 0.72 ADRB1 (0.63) HTR1AADRB2ADRB1ADRB3CYP1A2
SCHEMBL11337761 0.72 ADRB2 (0.51) HTR1AADRA2AADRB2ADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4215134-A B-RECEPTOR BLOCKING AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1980-07-29 US claimed
EP-0003298-B1 4-HYDROXY-2-BENZIMIDAZOLIN-THION DERIVATIVES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM Roche Diagnostics GmbH (DE) 1981-03-25 EP disclosed
US-4215134-A B-RECEPTOR BLOCKING AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1980-07-29 US disclosed