SCHEMBL11340443

SCHEMBL11340443

CCOc1nc2cccc(C)c2s1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ELANE P08246 1/20 0.42
KDM4E B2RXH2 1/20 0.38
MAPK1 P28482 1/20 0.38
HSD17B10 Q99714 1/20 0.38
F2RL3 Q96RI0 1/20 0.37
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 1/20 0.36
ACACB O00763 6/20 0.35
PTGS1 P23219 3/20 0.35
PTGS2 P35354 3/20 0.35
TLR8 Q9NR97 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11206376 0.82 PSMB8 (0.47) F2RL3HSP90AA1HSP90AB1KMT2AALDH1A1
SCHEMBL11347104 0.80 HSD17B10 (0.38) ELANEKDM4EMAPK1HSD17B10KMT2A
SCHEMBL9843032 0.74 CYP3A4 (0.39) ELANEKDM4EF2RL3KMT2AALDH1A1
SCHEMBL6842459 0.74 PTGS1 (0.58) KDM4EMAPK1F2RL3MEN1KMT2A
SCHEMBL12344033 0.74 TLR8 (0.46) KDM4EMAPK1F2RL3HSP90AA1HSP90AB1
SCHEMBL11216904 0.73 ALDH1A1 (0.53) KDM4EMAPK1HSD17B10F2RL3MEN1
SCHEMBL7958840 0.72 RAB9A (0.49) KDM4EHSD17B10ALDH1A1TLR8
SCHEMBL31063715 0.72 RAB9A (0.49) KDM4EHSD17B10ALDH1A1TLR8
SCHEMBL18026590 0.70 ACACB (0.47) KDM4EHSD17B10KMT2AACACB
SCHEMBL289210 0.69 SMN1; SMN2 (0.56) MAPK1HSD17B10HSP90AA1HSP90AB1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0039818-A1 Substituted 2-(3H)-benzothiazolones, processes for their preparation, their utilization in the preparation of medicines and medicines containing them Dr. Karl Thomae GmbH (DE) 1981-11-18 EP disclosed